SCHEMBL29862136

SCHEMBL29862136

CC(C)(C)OC(=O)N1C[C@@H](CCC(N[S+]([O-])C(C)(C)C)c2ccc(Br)cn2)CC1(C)C

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.35
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
FPR3 P25089 3/20 0.32
FPR2 P25090 3/20 0.32
CPB2 Q96IY4 1/20 0.32
POLB P06746 1/20 0.31
RORC P51449 2/20 0.31
IDO1 P14902 1/20 0.30
TDO2 P48775 1/20 0.30
ERBB2 P04626 1/20 0.30
EPHA2 P29317 1/20 0.30
KDR P35968 1/20 0.30
EPHB4 P54760 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23006414 1.00 DGAT1 (0.35) DGAT1NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL23006415 1.00 DGAT1 (0.35) DGAT1NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL23005972 0.90 HSD11B1 (0.33)
SCHEMBL23006297 0.90 SMN1; SMN2 (0.33) SMN1; SMN2CPB2ERBB2EPHA2KDR
SCHEMBL22982261 0.90 NPC1 (0.34) NPC1ALDH1A1RAB9ASMN1; SMN2POLB
SCHEMBL23005993 0.88 AAK1 (0.31) FPR3FPR2IDO1TDO2
SCHEMBL29862239 0.88 AAK1 (0.31) FPR3FPR2IDO1TDO2
SCHEMBL23005999 0.88 AAK1 (0.31) FPR3FPR2IDO1TDO2
SCHEMBL29862207 0.87 ADORA2B (0.36)
SCHEMBL28771552 0.87 ADORA2B (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220313698-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED 2022-10-06 US disclosed
EP-4013759-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR Vertex Pharmaceuticals Incorporated (US) 2022-06-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220313698-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR CFTR, SCNN1G, SCNN1B DGAT1 544/4885NPC1 271/4885ALDH1A1 3972/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.