SCHEMBL29862289

SCHEMBL29862289

O=C(c1cc(Cc2ccccc2)c(F)nc1F)N1CCOCC1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
TSHR P16473 4/20 0.54
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
GAA P10253 1/20 0.49
PLAUR Q03405 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 2/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
LMNA P02545 1/20 0.47
CNR1 P21554 2/20 0.46
HSP90AA1 P07900 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.44
FKBP1A P62942 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22982840 1.00 ALDH1A1 (0.54) ALDH1A1TSHRHTTSMN1; SMN2GAA
SCHEMBL22982237 0.78 PTPN1 (0.50) TSHRHSP90AA1
SCHEMBL3379273 0.74 ALDH1A1 (0.54) ALDH1A1TSHRHTTSMN1; SMN2GAA
SCHEMBL28771465 0.70 SSTR4 (0.39)
SCHEMBL7121916 0.69 SMN1; SMN2 (0.77) ALDH1A1TSHRHTTSMN1; SMN2GAA
SCHEMBL4473338 0.69 HSD17B10 (0.61) ALDH1A1TSHRHTTSMN1; SMN2GAA
SCHEMBL20387265 0.69 HTT (0.67) ALDH1A1TSHRHTTSMN1; SMN2GAA
SCHEMBL23309717 0.67 TSHR (0.54) ALDH1A1TSHRHTTSMN1; SMN2GAA
SCHEMBL20267430 0.67 GAA (0.73) ALDH1A1TSHRHTTSMN1; SMN2GAA
SCHEMBL14511637 0.67 PIN1 (0.50) ALDH1A1TSHRHTTSMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4013759-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR Vertex Pharmaceuticals Incorporated (US) 2022-06-22 EP disclosed