SCHEMBL2986594

SCHEMBL2986594

Cc1cc2c(B3OC(C)(C)C(C)(C)O3)ccnc2n1S(=O)(=O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 9/20 0.42
PIK3C3 Q8NEB9 1/20 0.38
HTR6 P50406 3/20 0.36
SRC P12931 2/20 0.36
BRD4 O60885 1/20 0.35
CYP2C19 P33261 1/20 0.34
GAA P10253 1/20 0.33
CCKAR P32238 1/20 0.33
LATS1 O95835 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16908341 0.91 PTGDR2 (0.40) PTGDR2CYP2C19GAALATS1NPSR1
SCHEMBL4602394 0.90 PTGDR2 (0.39) PTGDR2PIK3C3HTR6SRCBRD4
SCHEMBL30361980 0.88 PTGDR2 (0.38) PTGDR2PIK3C3HTR6SRCCYP2C19
SCHEMBL26103824 0.88 PTGDR2 (0.38) PTGDR2PIK3C3HTR6SRCCYP2C19
SCHEMBL15644711 0.87 PIK3C3 (0.41) PTGDR2PIK3C3HTR6SRCCYP2C19
SCHEMBL29514126 0.87 PTGDR2 (0.37) PTGDR2PIK3C3HTR6SRCCYP2C19
SCHEMBL4318668 0.87 PTGDR2 (0.37) PTGDR2PIK3C3HTR6SRCCYP2C19
SCHEMBL26720227 0.87 PTGDR2 (0.37) PTGDR2PIK3C3HTR6SRCCYP2C19
SCHEMBL13981488 0.85 PTGDR2 (0.38) PTGDR2PIK3C3HTR6SRCBRD4
SCHEMBL15646942 0.85 PTGDR2 (0.38) PTGDR2PIK3C3HTR6SRCCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250243196-A1 CITRON KINASE INHIBITORS THE CLEVELAND CLINIC FOUNDATION 2025-07-31 US disclosed
US-20230322772-A1 AZAINDOLYLPYRIDONE AND DIAZAINDOLYLPYRIDONE COMPOUNDS SPRINT BIOSCIENCE AB (SE) 2023-10-12 US disclosed
US-11498919-B2 Azaindolylpyridone and diazaindolylpyridone compounds SPRINT BIOSCIENCE AB (SE) 2022-11-15 US disclosed
WO-2022216717-A1 CITRON KINASE INHIBITORS THE CLEVELAND CLINIC FOUNDATION (US) 2022-10-13 WO disclosed
EP-4001278-A1 AZAINDOLYLPYRIDONE AND DIAZAINDOLYLPYRIDONE COMPOUNDS Sprint Bioscience AB (SE) 2022-05-25 EP disclosed
EP-3672967-B1 AZAINDOLYLPYRIDONE AND DIAZAINDOLYLPYRIDONE COMPOUNDS SPRINT BIOSCIENCE AB (SE) 2021-10-06 EP disclosed
US-20210122745-A1 AZAINDOLYLPYRIDONE AND DIAZAINDOLYLPYRIDONE COMPOUNDS SPRINT BIOSCIENCE AB (SE) 2021-04-29 US disclosed
EP-3129372-B1 AZAQUINAZOLINE INHIBITORS OF ATYPICAL PROTEIN KINASE C CANCER RESEARCH TECH LTD (GB) 2020-12-16 EP disclosed
EP-3129372-B1 AZAQUINAZOLINE INHIBITORS OF ATYPICAL PROTEIN KINASE C CANCER RESEARCH TECH LTD (GB) 2020-12-16 EP disclosed
EP-2900666-B1 AZAQUINAZOLINE INHIBITORS OF ATYPICAL PROTEIN KINASE C CANCER RESEARCH TECH LTD (GB) 2020-11-04 EP disclosed
US-20100035917-A1 PYRROLO[2,3-B]PYRIDIN-4-YL-BENZENESULFONAMIDE COMPOUNDS AS 1KK2 INHIBITORS GLAXO GROUP LIMITED (GB) 2010-02-11 US disclosed
WO-2008145688-A2 PYRROLOPYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS MEDICAMENTS GLAXO GROUP LIMITED (GB) 2008-12-04 WO disclosed
WO-2008145688-A2 PYRROLOPYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS MEDICAMENTS GLAXO GROUP LIMITED (GB) 2008-12-04 WO disclosed
US-20080176891-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-07-24 US disclosed
US-20080176891-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-07-24 US disclosed
US-20080176891-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-07-24 US disclosed
US-20080146606-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-06-19 US disclosed
US-20080146606-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-06-19 US disclosed
US-20080146606-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-06-19 US disclosed
WO-2008034860-A1 PYRROLO[2, 3-B]PYRIDIN-4-YL-BENZENESULFONAMIDE COMPOUNDS AS IKK2 INHIBITORS GLAXO GROUP LIMITED (GB) 2008-03-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230322772-A1 AZAINDOLYLPYRIDONE AND DIAZAINDOLYLPYRIDONE COMPOUNDS AZI2, IAPP, ZFX PTGDR2 498/4885PIK3C3 1407/4885HTR6 1633/4885
US-20210122745-A1 AZAINDOLYLPYRIDONE AND DIAZAINDOLYLPYRIDONE COMPOUNDS AZI2, IAPP, ZFX PTGDR2 498/4885PIK3C3 1407/4885HTR6 1633/4885
US-20080176891-A1 NOVEL COMPOUNDS NFKBIA, IKBKG, IKBKE PTGDR2 1284/4885PIK3C3 308/4885HTR6 4688/4885
US-20100035917-A1 PYRROLO[2,3-B]PYRIDIN-4-YL-BENZENESULFONAMIDE COMPOUNDS AS 1KK2 INHIBITORS PLK2, PDXK, MAP4K2 PTGDR2 2018/4885PIK3C3 548/4885HTR6 3710/4885
US-20080146606-A1 NOVEL COMPOUNDS NFKBIA, IKBKG, IKBKE PTGDR2 1284/4885PIK3C3 308/4885HTR6 4688/4885
US-20250243196-A1 CITRON KINASE INHIBITORS CHEK2, CILK1, DCK PTGDR2 3503/4885PIK3C3 734/4885HTR6 3372/4885
US-11498919-B2 Azaindolylpyridone and diazaindolylpyridone compounds AZI2, IAPP, ZFX PTGDR2 498/4885PIK3C3 1407/4885HTR6 1633/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.