SCHEMBL298748

SCHEMBL298748

NC(=O)c1ccc(C2(S(=O)(=O)O)CCCCC2)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 7/20 0.41
PAK1 Q13153 7/20 0.41
KDR P35968 3/20 0.41
NEK2 P51955 3/20 0.41
RIPK2 O43353 2/20 0.41
RAF1 P04049 2/20 0.41
MAP2K2 P36507 2/20 0.41
TGFBR2 P37173 2/20 0.41
MAP2K1 Q02750 2/20 0.41
TNK2 Q07912 2/20 0.41
MAP2K5 Q13163 2/20 0.41
PTK6 Q13882 2/20 0.41
NEK11 Q8NG66 2/20 0.41
MAP3K20 Q9NYL2 2/20 0.41
MAP4K5 Q9Y4K4 2/20 0.41
PLK4 O00444 2/20 0.41
AURKA O14965 2/20 0.41
ABL1 P00519 2/20 0.41
LCK P06239 2/20 0.41
FYN P06241 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298126 0.99 BRAF (0.42) BRAFPAK1KDRNEK2RIPK2
SCHEMBL297099 0.95 BRAF (0.43) BRAFPAK1KDRNEK2RIPK2
SCHEMBL298502 0.89 PAK1 (0.39) BRAFPAK1KDRNEK2RIPK2
SCHEMBL298555 0.89 CYP2C19 (0.41) BRAFPAK1KDRNEK2RIPK2
SCHEMBL297910 0.88 CYP2C19 (0.41) BRAFPAK1KDRNEK2RIPK2
SCHEMBL299063 0.88 PAK1 (0.40) BRAFPAK1KDRNEK2RIPK2
SCHEMBL299342 0.87 AAK1 (0.38) PAK1PTK6MAP3K20MAP4K5FES
SCHEMBL297236 0.86 AAK1 (0.39) PAK1KDRNEK2PTK6MAP3K20
SCHEMBL299489 0.83 PAK1 (0.49) PAK1TNIKPDPK1PAK4
SCHEMBL298746 0.82 CAMKK2 (0.57) PAK1KDRNEK2PLK4AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427433-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS Plexxikon, Inc. (US) 2012-03-14 EP disclosed