SCHEMBL299342

SCHEMBL299342

COc1cnc2[nH]cc(C(=O)c3cc(C(N)=O)ccc3C3(S(=O)(=O)O)CCCCC3)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.38
PAK1 Q13153 6/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
MAP3K11 Q16584 1/20 0.35
AXL P30530 3/20 0.33
CAMKK2 Q96RR4 2/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
DYRK1A Q13627 2/20 0.33
CLK1 P49759 1/20 0.33
DCLK1 O15075 1/20 0.33
DYRK3 O43781 1/20 0.33
ROCK2 O75116 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
EGFR P00533 1/20 0.33
NTRK1 P04629 1/20 0.33
CDK1 P06493 1/20 0.33
FES P07332 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL297236 0.99 AAK1 (0.39) AAK1PAK1MTNR1AMTNR1BMAP3K11
SCHEMBL298555 0.89 CYP2C19 (0.41) AAK1PAK1MAP3K11AXLCAMKK2
SCHEMBL297910 0.88 CYP2C19 (0.41) AAK1PAK1MAP3K11AXLCAMKK2
SCHEMBL298502 0.87 PAK1 (0.39) PAK1MAP3K11AXLCAMKK2CYP2C9
SCHEMBL298748 0.87 BRAF (0.41) PAK1AXLCYP2C9DYRK1ACLK1
SCHEMBL298126 0.86 BRAF (0.42) PAK1MAP3K11AXLCYP2C9DYRK1A
SCHEMBL299063 0.86 PAK1 (0.40) PAK1MAP3K11AXLCAMKK2CYP2C9
SCHEMBL299489 0.83 PAK1 (0.49) PAK1MKNK2
SCHEMBL297099 0.82 BRAF (0.43) PAK1MAP3K11AXLCAMKK2CYP2C9
SCHEMBL298746 0.82 CAMKK2 (0.57) AAK1PAK1MAP3K11AXLCAMKK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427433-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS Plexxikon, Inc. (US) 2012-03-14 EP disclosed