SCHEMBL29883010

SCHEMBL29883010

COc1cc2nccc(Oc3ccc(N(C(=O)C4(C(N)=O)CC4)c4ccc(F)cc4)cc3)c2cc1OC

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 11/20 0.66
AXL P30530 9/20 0.66
AURKB Q96GD4 4/20 0.66
KDR P35968 3/20 0.66
MERTK Q12866 3/20 0.66
FLT1 P17948 3/20 0.66
FLT3 P36888 2/20 0.66
AURKA O14965 1/20 0.66
RIPK2 O43353 1/20 0.66
ABCB11 O95342 1/20 0.66
ABL1 P00519 1/20 0.66
EGFR P00533 1/20 0.66
ERBB2 P04626 1/20 0.66
NTRK1 P04629 1/20 0.66
LCK P06239 1/20 0.66
PGR P06401 1/20 0.66
LYN P07948 1/20 0.66
RET P07949 1/20 0.66
CHRM2 P08172 1/20 0.66
HCK P08631 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL372017 1.00 MET (0.66) METAXLAURKBKDRMERTK
Pyruvate SCHEMBL29195420 0.96 MET (0.61) METAXLAURKBKDRMERTK
SCHEMBL31105630 0.94 MET (0.67) METAXLAURKBKDRMERTK
SCHEMBL28694985 0.94 MET (0.62) METAXLAURKBKDRMERTK
Glutarate SCHEMBL29195414 0.93 MET (0.58) METAXLAURKBKDRMERTK
SCHEMBL29453833 0.93 AXL (0.57) METAXLAURKBKDRMERTK
SCHEMBL22750248 0.93 AXL (0.57) METAXLAURKBKDRMERTK
SCHEMBL21201003 0.93 AXL (0.57) METAXLAURKBKDRMERTK
SCHEMBL410634 0.92 MET (0.58) METAXLAURKBKDRMERTK
SCHEMBL371952 0.92 AURKB (0.58) METAXLAURKBKDRMERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122036603-A Preparation method of anti-tumor drug cabatinib 新乡学院 2026-05-15 CN disclosed
US-20250333480-A1 FUSION MOLECULES AND USES THEREOF FOUNDATION MEDICINE, INC. (US) 2025-10-30 US disclosed
US-20250161276-A1 DRUG COMBINATIONS AND METHODS OF TREATING OVARIAN CANCER Pattern Computer, Inc. 2025-05-22 US disclosed
EP-4479047-A1 DRUG COMBINATIONS AND METHODS OF TREATING OVARIAN CANCER Pattern Computer, Inc. (US) 2024-12-25 EP disclosed
CN-118984704-A Pharmaceutical combinations and methods for treating ovarian cancer 帕特恩电脑公司 2024-11-19 CN disclosed
US-20240366608-A1 PHARMACEUTICAL COMBINATIONS OF SOS1 INHIBITORS FOR TREATING AND/OR PREVENTING CANCER LUPIN LIMITED (IN) 2024-11-07 US disclosed
EP-4313048-A1 PROCESS FOR PREPARATION OF CABOZANTINIB Biocon Limited (IN) 2024-02-07 EP disclosed
WO-2023234222-A1 METHOD FOR DETERMINING EFFECTIVENESS OF CANCER TREATMENT USING RET KINASE INHIBITOR 国立研究開発法人国立がん研究センター 2023-12-07 WO disclosed
CN-113164480-B Pharmaceutical composition for treating diffuse gastric cancer 学校法人金泽医科大学 2023-11-28 CN disclosed
WO-2023222946-A1 PROCESS FOR THE PREPARATION OF CABOZANTINIB FERMION OY (FI) 2023-11-23 WO disclosed
CN-116723843-A Pharmaceutical combination of SOS1 inhibitors for the treatment and/or prevention of cancer 鲁宾有限公司 2023-09-08 CN disclosed
WO-2023159184-A1 DRUG COMBINATIONS AND METHODS OF TREATING OVARIAN CANCER Pattern Computer, Inc. (US) 2023-08-24 WO disclosed
WO-2022201079-A1 PROCESS FOR PREPARATION OF CABOZANTINIB BIOCON LIMITED (IN) 2022-09-29 WO disclosed
WO-2022182982-A1 METHODS FOR TREATING C-KIT KINASE MEDIATED DISEASES AND DISORDERS USING A SELECTIVE C-KIT KINASE INHIBITOR THIRD HARMONIC BIO, INC. (US) 2022-09-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250161276-A1 DRUG COMBINATIONS AND METHODS OF TREATING OVARIAN CANCER TP53, TOP2A, BRCA1 MET 79/4885AXL 2912/4885AURKB 267/4885
US-20240366608-A1 PHARMACEUTICAL COMBINATIONS OF SOS1 INHIBITORS FOR TREATING AND/OR PREVENTING CANCER NRAS, KRAS, PRMT1 MET 48/4885AXL 449/4885AURKB 1401/4885
US-20250333480-A1 FUSION MOLECULES AND USES THEREOF RPS27A, CD2BP2, FGB MET 714/4885AXL 909/4885AURKB 1445/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.