SCHEMBL29888461

SCHEMBL29888461

c1ccc2c(c1)oc1cc(N3CCOCC3)ccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.56
PRKDC P78527 7/20 0.54
ACE P12821 1/20 0.54
ECE1 P42892 1/20 0.54
NPC1 O15118 5/20 0.52
RAB9A P51151 5/20 0.52
ALDH1A1 P00352 4/20 0.52
TP53 P04637 3/20 0.52
KDM4E B2RXH2 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
LMNA P02545 2/20 0.50
MEN1 O00255 4/20 0.48
MAPT P10636 4/20 0.48
KMT2A Q03164 4/20 0.48
HCRTR1 O43613 1/20 0.48
ATM Q13315 2/20 0.46
AHR P35869 1/20 0.46
CYP1A2 P05177 1/20 0.46
HTT P42858 1/20 0.46
LGMN Q99538 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29887322 0.83 HTR3A (0.53) NPC1RAB9AKDM4EMAPTAHR
SCHEMBL1938064 0.82 SLC16A3 (0.51) PRKDCACEECE1NPC1RAB9A
SCHEMBL19642427 0.78 MAOA (0.55) PRKDCNPC1RAB9AALDH1A1TP53
SCHEMBL2400184 0.77 PRKDC (0.51) PRKDCNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL14802157 0.74 PRKDC (0.50) TSHRPRKDCACEECE1NPC1
SCHEMBL5454434 0.74 MGAM (0.63) PRKDCACEECE1ALDH1A1KDM4E
SCHEMBL22742604 0.73 MAPT (0.57) TSHRPRKDCNPC1RAB9AALDH1A1
SCHEMBL22741398 0.73 MAPT (0.57) TSHRPRKDCNPC1RAB9AALDH1A1
SCHEMBL29886896 0.73 CHRNA7 (0.54) NPC1RAB9AALDH1A1KDM4ESMN1; SMN2
SCHEMBL24270394 0.73 KDM4E (0.60) PRKDCALDH1A1TP53KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114981251-B Dibenzofuran derivative cathepsin K inhibitor and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2023-11-21 CN disclosed
CN-114981251-A Diphenyl furan derivative cathepsin K inhibitor and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2022-08-30 CN disclosed