SCHEMBL14802157

SCHEMBL14802157

Cc1cc(N2CCOCC2)cc2oc3ccccc3c(=O)c12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 10/20 0.50
ACE P12821 1/20 0.50
ECE1 P42892 1/20 0.50
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAOA P21397 2/20 0.46
MGAM O43451 1/20 0.46
GAA P10253 1/20 0.46
SI P14410 1/20 0.46
MGAM2 Q2M2H8 1/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
HCRTR1 O43613 1/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
TSHR P16473 1/20 0.46
ATM Q13315 1/20 0.44
KIF11 P52732 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5454434 0.85 MGAM (0.63) PRKDCACEECE1KDM4EALDH1A1
SCHEMBL14802159 0.77 PRKDC (0.52) PRKDCKDM4EALDH1A1GAANPC1
SCHEMBL6895175 0.75 MAOA (0.57) KDM4EALDH1A1MAOAMGAMGAA
SCHEMBL14802143 0.75 PRKDC (0.52) PRKDCMAOAMGAMGAASI
SCHEMBL29888461 0.74 TSHR (0.56) PRKDCACEECE1KDM4EALDH1A1
SCHEMBL9837650 0.73 MGAM (0.72) KDM4EALDH1A1MAOAMGAMGAA
SCHEMBL1938064 0.72 SLC16A3 (0.51) PRKDCACEECE1KDM4EALDH1A1
SCHEMBL5440694 0.72 PRKDC (0.55) PRKDCACEKDM4EALDH1A1MAOA
SCHEMBL1794501 0.71 MAOA (0.63) KDM4EALDH1A1MAOAMGAMGAA
SCHEMBL18949722 0.71 AHR (0.57) KDM4EALDH1A1GAANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8404681-B2 Xanthones, thioxanthones and acridinones as DNA-PK inhibitors LUITPOLD PHARMACEUTICALS, INC. (US) 2013-03-26 US disclosed