SCHEMBL299482

SCHEMBL299482

FC(F)(F)c1nnc(-c2ccc(-c3cc4ccccc4s3)s2)s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.38
HSD17B1 P14061 1/20 0.38
HSD17B2 P37059 1/20 0.38
CYP19A1 P11511 1/20 0.37
ERN1 O75460 2/20 0.35
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
CA1 P00915 2/20 0.34
CA9 Q16790 2/20 0.34
CA2 P00918 1/20 0.34
NQO1 P15559 1/20 0.34
NQO2 P16083 1/20 0.34
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
CA12 O43570 1/20 0.33
IKBKB O14920 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5148513 0.76 APP (0.57) APPHSD17B1HSD17B2CYP19A1ERN1
SCHEMBL27651550 0.76 APP (0.57) APPHSD17B1HSD17B2CYP19A1ERN1
SCHEMBL26500221 0.74 APP (0.45) APPHSD17B1HSD17B2CYP19A1ERN1
SCHEMBL298901 0.74 KDM4E (0.46) ALDH1A1
SCHEMBL290560 0.72 BCL2L1 (0.40) APPHSD17B1HSD17B2CYP19A1ERN1
SCHEMBL290274 0.72 RAB9A (0.59) APPCYP19A1ALDH1A1
SCHEMBL29732980 0.71 APP (0.63) APPHSD17B1HSD17B2CYP19A1ERN1
SCHEMBL845603 0.71 APP (0.63) APPHSD17B1HSD17B2CYP19A1ERN1
SCHEMBL26744918 0.70 NPC1 (0.45) APPHSD17B1HSD17B2CYP19A1CA1
SCHEMBL288707 0.69 CYP19A1 (0.42) APPHSD17B1HSD17B2CYP19A1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed