SCHEMBL29890171

SCHEMBL29890171

COc1ccc(-c2cccc(=O)c(O)c2)cn1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 2/20 0.67
HSD17B2 P37059 2/20 0.67
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
ERN1 O75460 4/20 0.51
MKNK1 Q9BUB5 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
KEAP1 Q14145 1/20 0.48
NFE2L2 Q16236 1/20 0.48
PTGES2 Q9H7Z7 1/20 0.47
HDAC4 P56524 2/20 0.47
HDAC8 Q9BY41 2/20 0.47
HDAC2 Q92769 1/20 0.47
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
CTSA P10619 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23249824 1.00 HSD17B1 (0.67) HSD17B1HSD17B2CYP1A2CYP3A4CYP2C9
SCHEMBL23249859 0.82 FTO (0.51) HSD17B1HSD17B2PTGES2HDAC4HDAC8
SCHEMBL5673332 0.81 HSD17B1 (0.97) HSD17B1HSD17B2CYP1A2CYP3A4CYP2C9
SCHEMBL23249814 0.81 CNR1 (0.50) HSD17B1HSD17B2HDAC4HDAC8HDAC2
SCHEMBL23249811 0.80 HSD17B1 (0.42) HSD17B1HSD17B2ERN1MKNK1MKNK2
SCHEMBL29890188 0.80 HSD17B1 (0.42) HSD17B1HSD17B2ERN1MKNK1MKNK2
SCHEMBL29890034 0.78 HSD17B1 (0.41) HSD17B1HSD17B2CYP1A2CYP3A4CYP2C9
SCHEMBL23249818 0.78 HSD17B1 (0.41) HSD17B1HSD17B2CYP1A2CYP3A4CYP2C9
SCHEMBL29890158 0.77 FPR2 (0.50) PTGES2HDAC4HDAC8HDAC2PDGFRB
SCHEMBL23249841 0.77 FPR2 (0.50) PTGES2HDAC4HDAC8HDAC2PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4045025-A1 TROPOLONE DERIVATIVES AND TAUTOMERS THEREOF FOR IRON REGULATION IN ANIMALS Ambys Medicines, Inc. (US) 2022-08-24 EP disclosed