SCHEMBL29891703

SCHEMBL29891703

Cc1cccc(-c2noc(C3CCN(C(=O)OC(C)(C)C)CC3)n2)c1

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 18/20 0.60
CASP3 P42574 1/20 0.59
SENP7 Q9BQF6 1/20 0.59
SENP6 Q9GZR1 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23411281 1.00 GRM5 (0.60) GRM5CASP3SENP7SENP6
SCHEMBL1653518 0.89 TUBB4A (0.60)
SCHEMBL4423384 0.88 GPR119 (0.59)
SCHEMBL2901393 0.87 TUBB4A (0.58)
SCHEMBL20116734 0.87 L3MBTL1 (0.54) GRM5
SCHEMBL12580560 0.86 HCRTR1 (0.52) GRM5
SCHEMBL25171668 0.85 GRM5 (0.67) GRM5CASP3SENP7SENP6
SCHEMBL20116424 0.85 GRM5 (0.49) GRM5
SCHEMBL20116962 0.84 GRM5 (0.50) GRM5
SCHEMBL20116092 0.84 GRM5 (0.49) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119564686-A DGK alpha inhibitors as immune activation substituted aminoquinolones of (2) 拜耳公司 2025-03-07 CN disclosed
CN-119523983-A DGK alpha inhibitors as immune activation substituted aminoquinolones of (2) 拜耳公司 2025-02-28 CN disclosed
CN-119424429-A DGK alpha inhibitors as immune activation substituted aminoquinolones of (2) 拜耳公司 2025-02-14 CN disclosed
CN-115003665-B DGK alpha inhibitors as immune activation substituted aminoquinolones of (2) 拜耳公司 2024-11-08 CN disclosed
CN-115003665-A Substituted aminoquinolones as immunoactive DGK alpha inhibitors 拜耳公司 2022-09-02 CN disclosed