SCHEMBL2989339

SCHEMBL2989339

O=C1C=COC1C(=O)N1CCC2(CC1)N[C@@H](Cc1ccccc1)C(=O)N2Cc1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.35
MEN1 O00255 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
CCR5 P51681 4/20 0.34
CYP2D6 P10635 2/20 0.34
RIPK1 Q13546 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CHRM2 P08172 1/20 0.34
CYP3A4 P08684 1/20 0.34
HTT P42858 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
HDAC1 Q13547 3/20 0.32
HDAC6 Q9UBN7 3/20 0.32
HDAC8 Q9BY41 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2993037 0.89 HTT (0.33) CXCR3MEN1TSHRKMT2AALDH1A1
SCHEMBL3002193 0.88 CCR5 (0.40) CXCR3CCR5
SCHEMBL2989173 0.85 CCR5 (0.35) MEN1TSHRKMT2ACCR5CYP2D6
SCHEMBL3926088 0.83 CXCR3 (0.41) CXCR3CCR5CYP2D6RIPK1CHRM2
SCHEMBL1797763 0.81 CYP2D6 (0.51) CXCR3MEN1TSHRKMT2ACCR5
SCHEMBL4006029 0.81 CYP3A4 (0.55) MEN1TSHRKMT2ACYP2D6ALDH1A1
SCHEMBL1800751 0.81 CYP3A4 (0.55) MEN1TSHRKMT2ACYP2D6ALDH1A1
Hydrochloric Acid SCHEMBL1800654 0.80 CYP2D6 (0.50) CXCR3MEN1TSHRKMT2ACCR5
Hydrochloric Acid SCHEMBL1802546 0.80 CYP3A4 (0.54) MEN1TSHRKMT2ACYP2D6ALDH1A1
SCHEMBL3918198 0.80 GAA (0.41) CXCR3CCR5CYP2D6RIPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730147-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO[4,5]DECAN-2-ON COMPOUNDS FOR USE IN THE TREATMENT OF OBESITY GRUENENTHAL GMBH (DE) 2010-02-03 EP claimed