SCHEMBL3002193

SCHEMBL3002193

CCCCN1C(=O)C(Cc2ccccc2)NC12CCN(C(=O)C1OC=CC1=O)CC2

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.40
CXCR3 P49682 1/20 0.37
CXCR4 P61073 2/20 0.36
MMP1 P03956 1/20 0.34
MMP3 P08254 1/20 0.34
MMP9 P14780 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2989339 0.88 CXCR3 (0.35) CCR5CXCR3
SCHEMBL2993037 0.85 HTT (0.33) CXCR3
SCHEMBL1800591 0.82 CYP1A2 (0.47) CCR5
SCHEMBL1803393 0.82 CCR5 (0.49) CCR5
SCHEMBL1799903 0.79 CYP2D6 (0.47) CCR5CXCR3
SCHEMBL1798573 0.78 CCR5 (0.41) CCR5CXCR3CXCR4
SCHEMBL1799723 0.77 L3MBTL1 (0.42) CCR5CXCR3CXCR4
SCHEMBL1801308 0.77 CCR5 (0.49) CCR5
SCHEMBL2989173 0.76 CCR5 (0.35) CCR5
SCHEMBL1800826 0.75 CCR5 (0.39) CCR5CXCR3CXCR4MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730147-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO[4,5]DECAN-2-ON COMPOUNDS FOR USE IN THE TREATMENT OF OBESITY GRUENENTHAL GMBH (DE) 2010-02-03 EP claimed