SCHEMBL29907138

SCHEMBL29907138

Cn1cc(-c2nn(COCC[Si](C)(C)C)c3cc(Cl)c(Br)nc23)cn1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AXL P30530 3/20 0.35
DGAT1 O75907 3/20 0.34
PGK1 P00558 1/20 0.33
CNR2 P34972 2/20 0.31
CNR1 P21554 1/20 0.31
FGFR3 P22607 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23210897 1.00 AXL (0.35) AXLDGAT1PGK1CNR2CNR1
SCHEMBL19948747 0.83 DGAT1 (0.33) AXLDGAT1PGK1CNR2FGFR3
SCHEMBL1330040 0.79 AXL (0.46) AXLDGAT1
SCHEMBL23211133 0.79 CNR1 (0.34) CNR2CNR1
SCHEMBL29907197 0.79 CNR1 (0.34) CNR2CNR1
SCHEMBL29907034 0.78 DGAT1 (0.35) DGAT1
SCHEMBL23211119 0.78 DGAT1 (0.35) DGAT1
SCHEMBL19950254 0.77 CREBBP (0.33) AXLDGAT1PGK1
SCHEMBL30070423 0.77 CREBBP (0.33) AXLDGAT1PGK1
SCHEMBL22892770 0.77 MET (0.46) AXLPGK1FGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115835908-A Bicyclic heterocycles as FGFR inhibitors 因赛特公司 2023-03-21 CN disclosed
EP-4045151-A1 BICYCLIC HETEROCYCLES AS FGFR INHIBITORS Incyte Corporation (US) 2022-08-24 EP disclosed