SCHEMBL29909524

SCHEMBL29909524

CN(c1cccc(-c2nnc(C3CC3)o2)c1)c1nc2nnc(Cl)n2c2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
MAPT P10636 3/20 0.37
TNKS O95271 5/20 0.36
PARP2 Q9UGN5 5/20 0.36
PARP1 P09874 4/20 0.36
NR1H4 Q96RI1 4/20 0.36
BACE1 P56817 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
GAA P10253 1/20 0.35
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TP53 P04637 1/20 0.35
HTR4 Q13639 2/20 0.34
USP30 Q70CQ3 1/20 0.34
HSD11B1 P28845 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29909227 0.84 ABCG2 (0.34)
SCHEMBL29909333 0.82 ABCG2 (0.33)
SCHEMBL29909600 0.81 ABCG2 (0.32)
SCHEMBL29909714 0.81 MAP3K5 (0.33)
SCHEMBL29909542 0.81 ABCG2 (0.34)
SCHEMBL29909391 0.81 KDM4E (0.33) KDM4EMAPTTNKSPARP2PARP1
SCHEMBL29909736 0.80 GRM5 (0.33)
SCHEMBL23601014 0.79 MAPT (0.41) KDM4EMAPTTNKSPARP2PARP1
SCHEMBL29909431 0.77 ABCG2 (0.36) KDM4EMAPTALDH1A1
SCHEMBL29909406 0.77 ABCG2 (0.36) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12054490-B2 Diacylglycerol kinase modulating compounds GILEAD SCIENCES, INC. (US) 2024-08-06 US disclosed
CN-118324767-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-07-12 CN disclosed
EP-4081305-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS Carna Biosciences, Inc. (JP) 2022-11-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12054490-B2 Diacylglycerol kinase modulating compounds DGKG, DGKB, DGKK KDM4E 1748/4885MAPT 4206/4885TNKS 487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.