SCHEMBL29914724

SCHEMBL29914724

COc1ncc(-c2cccc(O)c2)cn1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FTO Q9C0B1 2/20 0.66
HSD17B1 P14061 9/20 0.64
HSD17B2 P37059 9/20 0.64
FYN P06241 4/20 0.51
BMPR1A P36894 1/20 0.51
TGFBR1 P36897 1/20 0.51
ACVRL1 P37023 1/20 0.51
ACVR1 Q04771 1/20 0.51
CYP3A4 P08684 3/20 0.50
CYP2C9 P11712 3/20 0.50
CYP1A2 P05177 1/20 0.49
CYP2C19 P33261 1/20 0.49
ABL1 P00519 1/20 0.46
FLT3 P36888 1/20 0.46
DYRK1A Q13627 1/20 0.44
DYRK1B Q9Y463 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28430998 1.00 FTO (0.66) FTOHSD17B1HSD17B2FYNBMPR1A
SCHEMBL23249859 0.80 FTO (0.51) FTOHSD17B1HSD17B2FYNDYRK1B
SCHEMBL13680543 0.80 FTO (0.50) FTOHSD17B1HSD17B2
SCHEMBL29431804 0.79 HSD17B1 (0.59) HSD17B1HSD17B2CYP3A4CYP2C9CYP1A2
SCHEMBL5673332 0.79 HSD17B1 (0.97) HSD17B1HSD17B2FYNBMPR1ATGFBR1
SCHEMBL23249732 0.79 FTO (1.00) FTOHSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL979785 0.79 MAP4K4 (0.65) FTOFYNCYP3A4ABL1FLT3
SCHEMBL15349707 0.78 PRKCI (0.51) FTOFYN
SCHEMBL30129857 0.77 FYN (0.60) HSD17B1HSD17B2FYNBMPR1ATGFBR1
SCHEMBL30129635 0.77 HSD17B1 (0.47) FTOHSD17B1HSD17B2FYNBMPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111094300-B Benzo-heteroaryl derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-09-16 CN disclosed