SCHEMBL2991540

SCHEMBL2991540

CCCNc1c(F)cccc1S(N)(=O)=O

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 9/20 0.45
ADRA2A P08913 1/20 0.40
ADRA2C P18825 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
CA1 P00915 6/20 0.38
CA2 P00918 6/20 0.38
CA9 Q16790 5/20 0.38
CA12 O43570 2/20 0.38
TRPA1 O75762 1/20 0.38
CISD1 Q9NZ45 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19121210 0.79 TRPA1 (0.44) TRPA1KMT2A
SCHEMBL3634671 0.75 HDAC1 (0.41) TRPA1KMT2A
SCHEMBL7354878 0.73 CA2 (0.59) PTGES2CA1CA2CA9CA12
SCHEMBL11660041 0.73 TRPA1 (0.43) TRPA1KMT2A
SCHEMBL30681712 0.72 PTGES2 (0.47) PTGES2CA1CA2CA9CA12
SCHEMBL30681713 0.72 PTGES2 (0.47) PTGES2CA1CA2CA9CA12
SCHEMBL17384694 0.72 PTGES2 (0.47) PTGES2CA1CA2CA9CA12
SCHEMBL18209561 0.71 PTGES2 (0.44) PTGES2CA1CA2CA9CA12
SCHEMBL29400968 0.70 HPGD (0.43) CA1CA2CA9CA12CISD1
SCHEMBL2778937 0.70 PTGES2 (0.44) PTGES2CA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2147915-B1 New cycloalkylated benzothiadiazine derivatives, method of preparing same and pharmaceutical compositions containing them SERVIER LAB (FR) 2010-09-15 EP disclosed