SCHEMBL29915641

SCHEMBL29915641

Nc1ccc(OCC2CCOC2)c(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.49
XDH P47989 5/20 0.41
IRAK4 Q9NWZ3 2/20 0.39
DHFR P00374 1/20 0.38
DCPS Q96C86 1/20 0.38
GRM4 Q14833 5/20 0.36
BRD4 O60885 2/20 0.36
TLR7 Q9NYK1 1/20 0.36
SCN8A Q9UQD0 1/20 0.35
FFAR2 O15552 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21652826 1.00 MCHR1 (0.49) MCHR1XDHIRAK4DHFRDCPS
SCHEMBL16650978 0.84 RIPK1 (0.41) MCHR1XDH
SCHEMBL21633961 0.83 MCHR1 (0.43) MCHR1XDHIRAK4GRM4BRD4
SCHEMBL30126151 0.83 MCHR1 (0.49) MCHR1XDHIRAK4DHFRDCPS
SCHEMBL21652799 0.83 CYP1A2 (0.43) MCHR1IRAK4BRD4
SCHEMBL30126942 0.83 MCHR1 (0.49) MCHR1XDHIRAK4DHFRDCPS
SCHEMBL30126836 0.83 MCHR1 (0.49) MCHR1XDHIRAK4DHFRDCPS
SCHEMBL23436644 0.80 MCHR1 (0.41) MCHR1XDHIRAK4GRM4BRD4
SCHEMBL21634036 0.78 CYP19A1 (0.42) MCHR1XDHIRAK4BRD4
SCHEMBL30127315 0.76 XDH (0.55) MCHR1XDHDHFRDCPSFFAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115716827-A Iminosulfones compound as bromodomain protein inhibitor, pharmaceutical composition and medical application thereof 正大天晴药业集团股份有限公司 2023-02-28 CN disclosed
CN-112424200-B Iminosulfones compound as bromodomain protein inhibitor, pharmaceutical composition and medical application thereof 正大天晴药业集团股份有限公司 2022-09-20 CN disclosed