SCHEMBL29919429

SCHEMBL29919429

CC(C)(C)OC(=O)N[C@@H](Cc1ccc(O[Si](C)(C)C(C)(C)C)cc1)CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.45
APP P05067 4/20 0.41
SCN9A Q15858 2/20 0.40
AKT1 P31749 1/20 0.39
PTPN1 P18031 2/20 0.39
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
HDAC8 Q9BY41 1/20 0.38
CTSS P25774 4/20 0.38
CTSK P43235 3/20 0.38
CCKAR P32238 1/20 0.38
CCKBR P32239 1/20 0.38
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25152858 1.00 ATM (0.45) ATMAPPSCN9AAKT1PTPN1
SCHEMBL27086909 0.89 KMT2A (0.40)
SCHEMBL27086914 0.89 KMT2A (0.40)
SCHEMBL13919601 0.87 ATM (0.49) ATMAPPSCN9AAKT1PTPN1
SCHEMBL8233202 0.87 ATM (0.49) ATMAPPAKT1CYP3A4
SCHEMBL13162709 0.87 ATM (0.51) ATMAPPSCN9AAKT1CTSS
SCHEMBL23375847 0.87 ATM (0.37) ATMAPPSCN9AAKT1CCKAR
SCHEMBL29688307 0.87 ATM (0.37) ATMAPPSCN9AAKT1CCKAR
SCHEMBL21447520 0.86 MC4R (0.37) ATMAPPSCN9AAKT1HDAC8
SCHEMBL29688277 0.86 MC4R (0.37) ATMAPPSCN9AAKT1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12168648-B2 Opioid receptor modulators EPIODYNE, INC. (US) 2024-12-17 US disclosed
US-20240092746-A1 OPIOID RECEPTOR MODULATORS EPIODYNE, INC. 2024-03-21 US disclosed
EP-4320105-A1 OPIOID RECEPTOR MODULATORS Epiodyne, Inc. (US) 2024-02-14 EP disclosed
US-11634396-B2 Opioid receptor modulators EPIODYNE, INC. (US) 2023-04-25 US disclosed
US-20220356157-A1 OPIOID RECEPTOR MODULATORS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-11-10 US disclosed
WO-2022216750-A1 OPIOID RECEPTOR MODULATORS EPIODYNE, INC. (US) 2022-10-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240092746-A1 OPIOID RECEPTOR MODULATORS OPRM1, OPRK1, OPRL1 ATM 4757/4885APP 3720/4885SCN9A 608/4885
US-12168648-B2 Opioid receptor modulators OPRM1, OPRK1, OPRL1 ATM 4757/4885APP 3720/4885SCN9A 608/4885
US-11634396-B2 Opioid receptor modulators OPRM1, OPRK1, OPRL1 ATM 4757/4885APP 3720/4885SCN9A 608/4885
US-20220356157-A1 OPIOID RECEPTOR MODULATORS OPRM1, OPRK1, OPRL1 ATM 4757/4885APP 3720/4885SCN9A 608/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.