SCHEMBL29922692

SCHEMBL29922692

Nc1ncc(-c2cc(N3CCOCC3)cc(S(=O)(=O)C3CCOC3)c2)c(C(F)(F)F)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 20/20 1.00
AKT1 P31749 13/20 1.00
MTOR P42345 8/20 0.74
PIK3C3 Q8NEB9 2/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21469886 1.00 PIK3CA (1.00) PIK3CAAKT1MTORPIK3C3
SCHEMBL23407481 0.87 PIK3CA (1.00) PIK3CAAKT1MTORPIK3C3
SCHEMBL21469765 0.87 PIK3CA (1.00) PIK3CAAKT1MTORPIK3C3
SCHEMBL21469838 0.86 PIK3CA (1.00) PIK3CAAKT1MTORPIK3C3
SCHEMBL23407499 0.86 PIK3CA (1.00) PIK3CAAKT1MTORPIK3C3
SCHEMBL29922694 0.86 PIK3CA (1.00) PIK3CAAKT1MTORPIK3C3
SCHEMBL21469824 0.85 PIK3CA (1.00) PIK3CAAKT1MTORPIK3C3
SCHEMBL29923012 0.85 PIK3CA (1.00) PIK3CAAKT1MTORPIK3C3
SCHEMBL21469827 0.85 PIK3CA (1.00) PIK3CAAKT1MTORPIK3C3
SCHEMBL29923044 0.85 PIK3CA (1.00) PIK3CAAKT1MTORPIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12637450-B2 Tri-substituted aryl and heteroaryl derivatives as modulators of PI3-kinase and autophagy pathways GLOBAL CANCER TECHNOLOGY INC. (US) 2026-05-26 US disclosed
US-20240327396-A1 TRI-SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES AS MODULATORS OF PI3-KINASE AND AUTOPHAGY PATHWAYS NEUROPORE THERAPIES, INC. (US) 2024-10-03 US disclosed
US-12049462-B2 Tri-substituted aryl and heteroaryl derivatives as modulators of PI3-kinase and autophagy pathways NEUROPORE THERAPIES, INC. (US) 2024-07-30 US disclosed
US-11492348-B2 Tri-substituted aryl and heteroaryl derivatives as modulators of PI3-kinase and autophagy pathways NEUROPORE THERAPIES, INC. (US) 2022-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11492348-B2 Tri-substituted aryl and heteroaryl derivatives as modulators of PI3-kinase and autophagy pathways ATG7, ULK1, BECN1 PIK3CA 31/4885AKT1 34/4885MTOR 4/4885
US-12637450-B2 Tri-substituted aryl and heteroaryl derivatives as modulators of PI3-kinase and autophagy pathways PIK3R4, PIK3R1, ATG7 PIK3CA 52/4885AKT1 32/4885MTOR 10/4885
US-20240327396-A1 TRI-SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES AS MODULATORS OF PI3-KINASE AND AUTOPHAGY PATHWAYS ATG7, ULK1, BECN1 PIK3CA 31/4885AKT1 34/4885MTOR 4/4885
US-12049462-B2 Tri-substituted aryl and heteroaryl derivatives as modulators of PI3-kinase and autophagy pathways ATG7, ULK1, BECN1 PIK3CA 31/4885AKT1 34/4885MTOR 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.