SCHEMBL29922728

SCHEMBL29922728

COC(=O)c1nnc(Cl)cc1NCc1ccc(OC)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 2/20 0.53
MAPT P10636 2/20 0.47
APLNR P35414 1/20 0.47
ALDH1A1 P00352 6/20 0.43
TSHR P16473 5/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ERBB2 P04626 1/20 0.43
PRKACA P17612 1/20 0.43
RPS6KB1 P23443 1/20 0.43
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43
IRAK1 P51617 1/20 0.43
RPS6KA3 P51812 1/20 0.43
ROCK1 Q13464 1/20 0.43
CDC42BPA Q5VT25 1/20 0.43
AURKB Q96GD4 1/20 0.43
CSNK1G3 Q9Y6M4 1/20 0.43
CYP1A2 P05177 4/20 0.43
CYP3A4 P08684 4/20 0.43
CYP2C19 P33261 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27007123 1.00 KDM4C (0.53) KDM4CMAPTAPLNRALDH1A1TSHR
SCHEMBL29552308 0.91 KDM4C (0.58) KDM4CMAPTAPLNRALDH1A1TSHR
SCHEMBL29937050 0.90 KDM4C (0.52) KDM4CMAPTAPLNRALDH1A1TSHR
SCHEMBL2135922 0.88 KDM4C (0.52) KDM4CMAPTAPLNRALDH1A1TSHR
SCHEMBL2599620 0.84 KDM4C (0.50) KDM4CMAPTAPLNRALDH1A1TSHR
SCHEMBL23015337 0.83 KDM4E (0.48) MAPTALDH1A1MEN1KMT2A
SCHEMBL25130656 0.83 APLNR (0.51) KDM4CMAPTAPLNRALDH1A1TSHR
SCHEMBL25131153 0.83 APLNR (0.54) KDM4CAPLNRALDH1A1TSHRERBB2
SCHEMBL30205616 0.83 APLNR (0.54) KDM4CAPLNRALDH1A1TSHRERBB2
SCHEMBL23486593 0.83 KDM4C (0.56) KDM4CMAPTAPLNRALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116096719-A Pyridazinylamino derivatives as ALK5 inhibitors 奇斯药制品公司 2023-05-09 CN disclosed
CN-110818641-B Pyridazine-3-formamide compound, preparation method and application thereof in medicine and pharmacology 北京诺诚健华医药科技有限公司 2022-10-14 CN disclosed