SCHEMBL29923201

SCHEMBL29923201

CCc1ccc(N)c(OC)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.34
NOS2 P35228 1/20 0.34
APOBEC3A P31941 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
ALDH1A1 P00352 6/20 0.33
PARP1 P09874 1/20 0.33
MBOAT4 Q96T53 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE3A Q14432 1/20 0.33
HEXA P06865 1/20 0.33
HEXB P07686 1/20 0.33
MAPT P10636 2/20 0.33
CASP1 P29466 2/20 0.33
CYP3A4 P08684 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
HSD17B10 Q99714 2/20 0.32
TSHR P16473 1/20 0.32
AURKA O14965 1/20 0.32
TTK P33981 1/20 0.32
AURKB Q96GD4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15148418 0.78 APOBEC3A (0.38) NOS3NOS2APOBEC3AAPOBEC3GALDH1A1
SCHEMBL13634487 0.78 PDE4B (0.39) APOBEC3AAPOBEC3GALDH1A1PDE4BPDE3A
SCHEMBL23343508 0.77 KCNH2 (0.36) ALDH1A1TDP1HRH2HRH3TLR7
SCHEMBL25010771 0.76 GRM4 (0.38) APOBEC3AAPOBEC3GPDE4BSMN1; SMN2KDM4E
SCHEMBL16802935 0.76 APOBEC3A (0.34) APOBEC3AAPOBEC3GALDH1A1PARP1PDE4B
SCHEMBL5155158 0.76 CHEK1 (0.44) ALDH1A1MAPTTDP1HSD17B10SMN1; SMN2
SCHEMBL2637242 0.75 PGK1 (0.49) MBOAT4TLR8TLR7
SCHEMBL13746013 0.74 NCF1 (0.42) NOS3NOS2ALDH1A1MAPTCASP1
SCHEMBL10399548 0.74 NOS3 (0.39) NOS3NOS2ALDH1A1PARP1HEXA
SCHEMBL21582525 0.73 MAPT (0.39) APOBEC3GALDH1A1MAPTCASP1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4334305-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2024-03-13 EP disclosed
WO-2022236101-A1 WDR5 INHIBITORS AND MODULATORS VANDERBILT UNIVERSITY (US) 2022-11-10 WO disclosed
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed