SCHEMBL29923343

SCHEMBL29923343

CCc1cc(C(=O)O)c2ncccc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.52
PDE4A P27815 1/20 0.50
ALDH1A1 P00352 4/20 0.49
LMNA P02545 3/20 0.46
ALOX12 P18054 1/20 0.46
EGLN1 Q9GZT9 4/20 0.44
KDM4E B2RXH2 5/20 0.42
TDP1 Q9NUW8 2/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
TET2 Q6N021 2/20 0.42
TET1 Q8NFU7 2/20 0.42
KDM6B O15054 1/20 0.42
KDM6A O15550 1/20 0.42
TET3 O43151 1/20 0.42
KDM4A O75164 1/20 0.42
KDM4B O94953 1/20 0.42
KDM5C P41229 1/20 0.42
KDM4D Q6B0I6 1/20 0.42
ALKBH5 Q6P6C2 1/20 0.42
FTO Q9C0B1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29923736 0.87 PARP1 (0.66) PARP1PDE4AALDH1A1EGLN1KDM4E
SCHEMBL29923860 0.84 PARP1 (0.49) PARP1PDE4AEGLN1TDP1MAPT
SCHEMBL22288232 0.82 PARP1 (0.44) PARP1PDE4AALDH1A1LMNAEGLN1
SCHEMBL21816294 0.80 PSMD14 (0.56) PARP1ALDH1A1LMNAALOX12EGLN1
SCHEMBL18484186 0.79 ALDH1A1 (0.47) PARP1PDE4AALDH1A1LMNAALOX12
SCHEMBL29923798 0.79 NPC1 (0.52) PDE4AALDH1A1LMNAEGLN1KDM4E
SCHEMBL29923816 0.79 EGLN1 (0.54) PARP1EGLN1KDM4EL3MBTL1TET2
SCHEMBL29923706 0.79 PARP1 (0.42) PARP1PDE4AALDH1A1LMNAEGLN1
SCHEMBL68215 0.78 ALDH1A1 (0.54) PARP1PDE4AALDH1A1LMNAALOX12
SCHEMBL686939 0.78 KDM4E (0.53) PARP1ALOX12KDM4ETDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-B1 WDR5 INHIBITORS AND MODULATORS UNIV VANDERBILT (US) 2024-03-20 EP disclosed
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed