SCHEMBL29923797

SCHEMBL29923797

COc1cc(COC2CC2)c2nccc(Br)c2c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GRM2 Q14416 1/20 0.34
HTR1A P08908 9/20 0.33
SLC6A4 P31645 8/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
NSD2 O96028 1/20 0.32
CASP6 P55212 1/20 0.32
CARM1 Q86X55 1/20 0.32
PRMT6 Q96LA8 1/20 0.32
EIF2AK2 P19525 1/20 0.31
GPR84 Q9NQS5 1/20 0.31
CCR1 P32246 1/20 0.30
CCR5 P51681 1/20 0.30
CCR8 P51685 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24916107 1.00 KDM4E (0.38) KDM4EL3MBTL1GRM2HTR1ASLC6A4
SCHEMBL24916497 0.95 KDM4E (0.41) KDM4EL3MBTL1GRM2HTR1ASLC6A4
SCHEMBL24915872 0.91 CARM1 (0.37) KDM4EL3MBTL1HTR1ASLC6A4CARM1
SCHEMBL24915807 0.84 KDM4E (0.38) KDM4EL3MBTL1HTR1AHSP90AA1HSP90AB1
SCHEMBL29923349 0.84 KDM4E (0.38) KDM4EL3MBTL1HTR1AHSP90AA1HSP90AB1
SCHEMBL24916031 0.83 KDM4E (0.36) KDM4EL3MBTL1SLC6A4HSP90AA1HSP90AB1
SCHEMBL29923321 0.80 NSD2 (0.38) KDM4EHTR1AHSP90AA1HSP90AB1NSD2
SCHEMBL24916137 0.80 NSD2 (0.38) KDM4EHTR1AHSP90AA1HSP90AB1NSD2
SCHEMBL24916038 0.79 KDM4E (0.40) KDM4EL3MBTL1HTR1ASLC6A4HSP90AA1
SCHEMBL24916306 0.79 CYP19A1 (0.38) KDM4EHSP90AA1HSP90AB1NSD2CASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed