SCHEMBL29923914

SCHEMBL29923914

CCOc1ccc2nc(C(=O)O)ccc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.55
ALDH1A1 P00352 5/20 0.55
SMN1; SMN2 Q16637 4/20 0.55
HSD17B10 Q99714 3/20 0.55
HPGD P15428 3/20 0.55
TSHR P16473 2/20 0.55
CYP1A2 P05177 1/20 0.55
AKR1C3 P42330 1/20 0.51
AKR1C2 P52895 1/20 0.51
MGAM O43451 1/20 0.47
RAB9A P51151 4/20 0.47
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
NCF1 P14598 1/20 0.46
NPC1 O15118 3/20 0.45
MAPT P10636 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
THRB P10828 1/20 0.45
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11054926 0.85 TP53 (0.54) TSHRTP53
SCHEMBL9945361 0.84 AKR1C3 (0.51) KDM4EALDH1A1SMN1; SMN2HSD17B10HPGD
SCHEMBL1993328 0.83 KDM4E (0.57) KDM4EALDH1A1SMN1; SMN2HSD17B10HPGD
SCHEMBL21864940 0.81 P4HTM (0.61) KDM4EALDH1A1HSD17B10HPGDCYP1A2
SCHEMBL2908071 0.79 KDM4E (0.59) KDM4EALDH1A1SMN1; SMN2HSD17B10HPGD
SCHEMBL6102490 0.79 AKR1C3 (0.51) KDM4EALDH1A1SMN1; SMN2HSD17B10HPGD
SCHEMBL28231529 0.76 SMN1; SMN2 (0.50) SMN1; SMN2HSD17B10CYP1A2MGAMRAB9A
SCHEMBL867738 0.76 KDM4E (0.66) KDM4ESMN1; SMN2TSHRAKR1C3AKR1C2
SCHEMBL9694076 0.76 KDM4E (0.54) KDM4EALDH1A1SMN1; SMN2HSD17B10HPGD
SCHEMBL31222310 0.75 ALDH1A1 (0.58) KDM4EALDH1A1SMN1; SMN2HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed