SCHEMBL29924260

SCHEMBL29924260

OC(COc1cccc(Br)c1I)c1ccc(Cl)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
GRIN2B Q13224 3/20 0.35
S1PR4 O95977 1/20 0.35
KCNH2 Q12809 2/20 0.35
KMT2A Q03164 1/20 0.35
HPGD P15428 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
SLC2A1 P11166 1/20 0.33
HRH1 P35367 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33
PPARA Q07869 1/20 0.33
NPC1 O15118 1/20 0.32
TSHR P16473 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29149893 1.00 ADRA2C (0.36) ADRA2CCYP1A2CYP2D6GRIN2BS1PR4
SCHEMBL29149840 0.88 KCNH2 (0.40) GRIN2BKCNH2KMT2AHPGDSMN1; SMN2
SCHEMBL29924274 0.88 KCNH2 (0.40) GRIN2BKCNH2KMT2AHPGDSMN1; SMN2
SCHEMBL29924223 0.87 KMT2A (0.38) CYP1A2KMT2ALMNAMAPT
SCHEMBL29150120 0.87 KMT2A (0.38) CYP1A2KMT2ALMNAMAPT
SCHEMBL29924357 0.78 APLNR (0.34) GRIN2BS1PR4KMT2AHPGDSMN1; SMN2
SCHEMBL29150016 0.78 APLNR (0.34) GRIN2BS1PR4KMT2AHPGDSMN1; SMN2
SCHEMBL24186460 0.74 KCNH2 (0.40) GRIN2BKCNH2KMT2AHPGDSMN1; SMN2
SCHEMBL29924532 0.73 S1PR4 (0.43) S1PR4KMT2AHPGDSMN1; SMN2ALDH1A1
SCHEMBL29924520 0.72 ALDH1A1 (0.47) KMT2AALDH1A1LMNAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117177970-A Polycyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-05 CN disclosed
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed