SCHEMBL29924291

SCHEMBL29924291

COC(=O)c1ccc2nc(CCl)n(CC3(CF)CC3)c2n1

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.35
PPARG P37231 2/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29924769 0.90 CYP1A2 (0.38) MAPT
SCHEMBL25004893 0.90 CYP1A2 (0.38) MAPT
SCHEMBL27237114 0.87 LMNA (0.32)
SCHEMBL30882773 0.87 LMNA (0.35) PTGER4PPARG
SCHEMBL25005199 0.87 LMNA (0.35) PTGER4PPARG
SCHEMBL29946034 0.80 ACSS2 (0.43)
SCHEMBL25340079 0.80 ACSS2 (0.43)
SCHEMBL30798199 0.78 TP53 (0.44) PTGER4MAPT
SCHEMBL31143242 0.77 MAPT (0.38) PTGER4PPARGMAPT
SCHEMBL31143304 0.77 MAPT (0.38) PTGER4PPARGMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117986264-A Benzo nitrogen-containing polycyclic derivative regulator and preparation method and application thereof 江苏豪森药业集团有限公司 2024-05-07 CN disclosed
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed