SCHEMBL29924720

SCHEMBL29924720

S=C(Nc1ccccc1)c1ccncc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.62
LMNA P02545 4/20 0.62
TDP1 Q9NUW8 1/20 0.62
HTT P42858 2/20 0.61
ALDH1A1 P00352 3/20 0.58
CA9 Q16790 2/20 0.58
CA1 P00915 1/20 0.58
GAA P10253 1/20 0.58
MAPT P10636 3/20 0.57
HPGD P15428 3/20 0.57
NPC1 O15118 4/20 0.56
RAB9A P51151 4/20 0.56
CYP3A4 P08684 2/20 0.56
CYP1A2 P05177 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
TAAR1 Q96RJ0 1/20 0.55
KMT2A Q03164 2/20 0.55
CCR6 P51684 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL557621 0.85 NPC1 (0.73) SMN1; SMN2LMNAHTTALDH1A1GAA
SCHEMBL10978008 0.85 NPC1 (0.71) SMN1; SMN2LMNAALDH1A1GAAMAPT
SCHEMBL28056929 0.83 ATG4B (0.59) SMN1; SMN2LMNATDP1HTTALDH1A1
SCHEMBL9317188 0.83 NPC1 (0.70) SMN1; SMN2LMNAHTTALDH1A1GAA
SCHEMBL9317189 0.83 NPC1 (0.70) SMN1; SMN2LMNAHTTALDH1A1GAA
SCHEMBL16566469 0.79 ALDH1A1 (0.74) SMN1; SMN2LMNATDP1HTTALDH1A1
Naphthalene SCHEMBL9316632 0.78 NPC1 (0.63) SMN1; SMN2LMNAHTTALDH1A1GAA
SCHEMBL10382103 0.78 GAA (0.64) SMN1; SMN2LMNAALDH1A1GAAMAPT
SCHEMBL11920080 0.77 SMN1; SMN2 (1.00) SMN1; SMN2LMNATDP1HTTALDH1A1
SCHEMBL28471166 0.76 NPC1 (0.61) SMN1; SMN2LMNAALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4288419-A1 1,3,4-OXADIAZOLE THIOCARBONYL COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME Chong Kun Dang Pharmaceutical Corp. (KR) 2023-12-13 EP disclosed
CN-117120421-A 1,3, 4-oxadiazole thiocarbonyl compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions containing the same 株式会社钟根堂 2023-11-24 CN disclosed
WO-2022215020-A1 1,3,4-OXADIAZOLE THIOCARBONYL COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2022-10-13 WO disclosed