SCHEMBL29930712

SCHEMBL29930712

C[Si](C)(C)CCOCn1nc(-c2ccccc2)c2cc(-c3ccc(O)cc3)cnc21

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
GSK3B P49841 1/20 0.38
MERTK Q12866 5/20 0.38
ESR1 P03372 6/20 0.37
USP7 Q93009 1/20 0.37
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
AXL P30530 2/20 0.34
TYRO3 Q06418 2/20 0.34
POLB P06746 1/20 0.34
DGAT1 O75907 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29930820 0.95 GSK3B (0.41) GSK3BMERTKMAPTNPC1AXL
SCHEMBL29930904 0.91 CLK1 (0.39) DYRK1ADYRK1BGSK3BMERTKESR1
SCHEMBL27215091 0.90 MERTK (0.39) MERTKESR1MAPTNPC1AXL
SCHEMBL29930818 0.88 HSD17B2 (0.39) DYRK1ADYRK1BNPC1DGAT1
SCHEMBL29930809 0.85 DGAT1 (0.37) DYRK1ADYRK1BMERTKESR1MAPT
SCHEMBL29930883 0.84 AXL (0.42) DYRK1AGSK3BMERTKMAPTAXL
SCHEMBL29930958 0.80 AXL (0.39) MERTKMAPTNPC1AXLTYRO3
SCHEMBL29930755 0.79 L3MBTL1 (0.40) MERTKNPC1
SCHEMBL29930865 0.77 DYRK1A (0.44) DYRK1ADYRK1BMERTKMAPTAXL
SCHEMBL29930517 0.76 PTPN11 (0.47) MERTKMAPTNPC1AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022235097-A1 PHARMACEUTICAL COMPOSITION CONTAINING NOVEL PYRAZOLO[3,4-B]PYRIDINE DERIVATIVE FOR PREVENTION OR TREATMENT OF METABOLIC DISEASE INCLUDING OBESITY AND DIABETES MELLITUS OR NONALCOHOLIC STEATOHEPATITIS 한국화학연구원 2022-11-10 WO disclosed