SCHEMBL29937282

SCHEMBL29937282

O=C1OCCc2ncncc21

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 1/20 0.38
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA9 Q16790 1/20 0.35
HTR1A P08908 2/20 0.32
DRD2 P14416 2/20 0.32
HTR2A P28223 2/20 0.32
ALDH1A1 P00352 2/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18013209 0.81 MAOA (0.36) CDC25BALDH1A1LMNATSHR
SCHEMBL30640315 0.81 MAOA (0.36) CDC25BALDH1A1LMNATSHR
SCHEMBL9538581 0.72
SCHEMBL15386166 0.72 CDC25B (0.38) CDC25BCA1CA2CA4CA9
SCHEMBL30443999 0.72 CDC25B (0.38) CDC25BCA1CA2CA4CA9
SCHEMBL15509407 0.72 TDP2 (0.45) CDC25B
SCHEMBL29448312 0.72 TDP2 (0.45) CDC25B
SCHEMBL29502224 0.69 GRM5 (0.47) CDC25BCA1CA2CA4CA9
SCHEMBL3224277 0.69 GRM5 (0.47) CDC25BCA1CA2CA4CA9
Hydrochloric Acid SCHEMBL31585763 0.68 GRM5 (0.46) CDC25BCA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4322954-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT Merck Sharp & Dohme LLC (US) 2024-02-21 EP disclosed
WO-2022221739-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT MERCK SHARP & DOHME CORP. (US) 2022-10-20 WO disclosed