SCHEMBL29937409

SCHEMBL29937409

O=c1ncc2nnccc2[nH]1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATAD2 Q6PL18 1/20 0.35
MAPKAPK2 P49137 1/20 0.33
RPS6KA3 P51812 1/20 0.33
CSNK2A1 P68400 1/20 0.33
PLK3 Q9H4B4 1/20 0.33
DAO P14920 1/20 0.32
PDE3B Q13370 3/20 0.32
PDE3A Q14432 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18035168 1.00 ATAD2 (0.35) ATAD2MAPKAPK2RPS6KA3CSNK2A1PLK3
SCHEMBL167012 0.74 ATAD2 (0.56) ATAD2DAOPDE3BPDE3A
SCHEMBL2898417 0.73 ATAD2 (0.54) ATAD2DAOPDE3BPDE3A
SCHEMBL29578870 0.72 PDE3B (0.46) MAPKAPK2RPS6KA3CSNK2A1PLK3PDE3B
SCHEMBL2811653 0.69 PKM (0.31)
SCHEMBL24558925 0.68 KDM4E (0.38) ATAD2MAPKAPK2RPS6KA3CSNK2A1PLK3
SCHEMBL30528447 0.67
SCHEMBL219125 0.67
SCHEMBL7051447 0.67 PDE3B (0.58) DAOPDE3BPDE3A
SCHEMBL27791126 0.66 ATAD2 (0.46) ATAD2DAOPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4322954-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT Merck Sharp & Dohme LLC (US) 2024-02-21 EP disclosed
WO-2022221739-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT MERCK SHARP & DOHME CORP. (US) 2022-10-20 WO disclosed