SCHEMBL29940543

SCHEMBL29940543

N#Cc1ccc2c(c1)Cc1c([nH]c3ccccc13)C2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 2/20 0.48
CDK1 P06493 2/20 0.48
CCNB1 P14635 2/20 0.48
GSK3B P49841 2/20 0.48
CCNB3 Q8WWL7 2/20 0.48
DRD2 P14416 7/20 0.46
DRD1 P21728 7/20 0.46
DRD5 P21918 7/20 0.46
DRD3 P35462 6/20 0.46
DRD4 P21917 5/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
GMNN O75496 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
ADRA1D P25100 1/20 0.46
CYP2C19 P33261 1/20 0.46
ADRA1A P35348 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20356899 0.86 MAPK10 (0.46) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL31737740 0.86 MAPK10 (0.46) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL23636196 0.80 DRD5 (0.64) DRD2DRD1DRD5DRD3DRD4
SCHEMBL30009136 0.78 MAPK10 (0.41) DRD2DRD3
SCHEMBL30569664 0.73 HTR2A (0.57) DRD2DRD1DRD5DRD3DRD4
SCHEMBL30569666 0.73 HTR2A (0.57) DRD2DRD1DRD5DRD3DRD4
SCHEMBL1120971 0.73 HTR2A (0.57) DRD2DRD1DRD5DRD3DRD4
SCHEMBL10019851 0.73 HTR2A (0.57) DRD2DRD1DRD5DRD3DRD4
SCHEMBL20356888 0.71 HTR6 (0.47) DRD2DRD1DRD5DRD3DRD4
SCHEMBL6739755 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115340523-B Compound with ALK inhibitory activity and preparation method and application thereof 盛世泰科生物医药技术(苏州)股份有限公司 2023-12-15 CN disclosed
WO-2022237813-A1 COMPOUND HAVING ALK INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 盛世泰科生物医药技术(苏州)有限公司 2022-11-17 WO disclosed
CN-115340523-A Compound with ALK inhibitory activity and preparation method and application thereof 盛世泰科生物医药技术(苏州)有限公司 2022-11-15 CN disclosed