SCHEMBL30009136

SCHEMBL30009136

C[Si](C)(C)C#Cc1ccc2c3c([nH]c2c1)Cc1ccc(C#N)cc1C3

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 2/20 0.41
RIPK1 Q13546 2/20 0.41
ALK Q9UM73 5/20 0.32
FLT3 P36888 3/20 0.32
DRD2 P14416 2/20 0.32
DRD3 P35462 2/20 0.32
PNMT P11086 1/20 0.32
CHEK1 O14757 2/20 0.32
CHEK2 O96017 1/20 0.32
ITK Q08881 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
CFB P00751 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20356899 0.80 MAPK10 (0.46) MAPK10RIPK1DRD2DRD3ITK
SCHEMBL31737740 0.80 MAPK10 (0.46) MAPK10RIPK1DRD2DRD3ITK
SCHEMBL30009067 0.78 ALK (0.46) ALKFLT3
SCHEMBL29940543 0.78 CCNB2 (0.48) DRD2DRD3
SCHEMBL30009089 0.67 FLT3 (0.36) ALKFLT3
SCHEMBL25183518 0.65 MAPK10 (0.47) MAPK10RIPK1ALKDRD2DRD3
SCHEMBL6849836 0.65 GABRA1 (0.37)
SCHEMBL5775576 0.65 CYP11B1 (0.43)
SCHEMBL9152103 0.65 MAPT (0.50) MAPK10RIPK1
SCHEMBL6739755 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237813-A1 COMPOUND HAVING ALK INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 盛世泰科生物医药技术(苏州)有限公司 2022-11-17 WO disclosed