SCHEMBL29951589

SCHEMBL29951589

O=Cc1c(Br)nn(-c2ccc(C(F)(F)F)cc2)c1Br

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.39
CYP2C9 P11712 3/20 0.39
PDPK1 O15530 1/20 0.38
ATM Q13315 1/20 0.37
HIF1A Q16665 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ENPP2 Q13822 1/20 0.35
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
SRC P12931 1/20 0.33
BRAF P15056 1/20 0.33
KDR P35968 1/20 0.33
HDAC3 O15379 1/20 0.33
ADAM17 P78536 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29955468 0.83 KMT2A (0.43) MAPTRAB9AL3MBTL1
SCHEMBL2562844 0.83 CA1 (0.37) PTGS2CYP2C9L3MBTL1PTGS1CYP2D6
SCHEMBL29953059 0.81 NPSR1 (0.47) PTGS2CYP2C9PDPK1HIF1AKDM4E
SCHEMBL2556063 0.80 PTGS1 (0.37) PTGS2MAPTRAB9AL3MBTL1PTGS1
SCHEMBL29953701 0.78 NPSR1 (0.47) PTGS2CYP2C9PDPK1KDM4ENPSR1
SCHEMBL2557923 0.76 CA1 (0.35) PTGS2PTGS1
SCHEMBL2558155 0.75 MAPT (0.46) PTGS2KDM4EMAPTRAB9APTGS1
SCHEMBL29951698 0.74 ALDH1A1 (0.37) CYP2C9KDM4EMAPTL3MBTL1CYP2D6
SCHEMBL2556085 0.73
SCHEMBL5904596 0.73 BRAF (0.43) PTGS2CYP2C9PDPK1ATMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed