SCHEMBL29953701

SCHEMBL29953701

O=Cc1c(-c2ccc(C(F)(F)F)cc2)nn(-c2ccccc2)c1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.47
KDM4E B2RXH2 2/20 0.47
LMNA P02545 2/20 0.42
ALDH1A1 P00352 1/20 0.42
GRM5 P41594 1/20 0.40
BRAF P15056 3/20 0.39
SRC P12931 2/20 0.39
KDR P35968 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KIF11 P52732 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
PTGER1 P34995 1/20 0.39
BACE1 P56817 1/20 0.38
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
PTGS2 P35354 2/20 0.37
CYP2C9 P11712 1/20 0.37
NPY5R Q15761 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29953059 0.95 NPSR1 (0.47) NPSR1KDM4ELMNAALDH1A1GRM5
SCHEMBL15332775 0.87 LMNA (0.40) NPSR1KDM4ELMNAALDH1A1MEN1
SCHEMBL29951388 0.86 ALDH1A1 (0.50) NPSR1LMNAALDH1A1MEN1KMT2A
SCHEMBL29953830 0.86 ALDH1A1 (0.59) NPSR1LMNAALDH1A1GRM5MEN1
SCHEMBL11726388 0.86 PTGS2 (0.46) NPSR1LMNAALDH1A1SRCMEN1
SCHEMBL15330588 0.85 POLB (0.52) NPSR1KDM4ELMNAALDH1A1BRAF
SCHEMBL11732622 0.83 NPSR1 (0.53) NPSR1KDM4ELMNASRCMEN1
SCHEMBL15331371 0.83 LMNA (0.46) NPSR1KDM4ELMNAALDH1A1MEN1
SCHEMBL15333698 0.80 POLB (0.46) NPSR1KDM4ELMNAALDH1A1BRAF
SCHEMBL2557352 0.80 CA1 (0.39) NPSR1LMNAALDH1A1GRM5BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed