SCHEMBL29953059

SCHEMBL29953059

O=Cc1c(-c2ccccc2)nn(-c2ccc(C(F)(F)F)cc2)c1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
GRM5 P41594 1/20 0.40
SRC P12931 1/20 0.39
BRAF P15056 1/20 0.39
KDR P35968 1/20 0.39
KIF11 P52732 1/20 0.39
BACE1 P56817 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
PTGS2 P35354 7/20 0.38
PTGS1 P23219 5/20 0.38
EPHX2 P34913 2/20 0.38
HIF1A Q16665 1/20 0.37
CYP2C9 P11712 1/20 0.37
PTGER1 P34995 1/20 0.36
NPY5R Q15761 1/20 0.36
PDPK1 O15530 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29953701 0.95 NPSR1 (0.47) NPSR1KDM4EALDH1A1LMNAGRM5
SCHEMBL29951388 0.86 ALDH1A1 (0.50) NPSR1ALDH1A1LMNACYP2C9NPY5R
SCHEMBL29953830 0.86 ALDH1A1 (0.59) NPSR1ALDH1A1LMNAGRM5PTGS1
SCHEMBL11726388 0.86 PTGS2 (0.46) NPSR1ALDH1A1LMNASRCCA1
SCHEMBL15333698 0.85 POLB (0.46) NPSR1KDM4EALDH1A1LMNASRC
SCHEMBL15332775 0.82 LMNA (0.40) NPSR1KDM4EALDH1A1LMNACA1
SCHEMBL29951589 0.81 PTGS2 (0.39) NPSR1KDM4ESRCBRAFKDR
SCHEMBL15330588 0.80 POLB (0.52) NPSR1KDM4EALDH1A1LMNASRC
SCHEMBL29954291 0.80 RXRA (0.38) NPSR1KDM4EALDH1A1LMNAPTGS2
SCHEMBL2556343 0.80 HTT (0.36) NPSR1KDM4EALDH1A1LMNAGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed