SCHEMBL29952086

SCHEMBL29952086

Nc1nc(C(F)(F)F)ccc1B(O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TKT P29401 1/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
P2RX7 Q99572 1/20 0.34
KCNH2 Q12809 3/20 0.33
MAP4K4 O95819 1/20 0.33
PIK3CA P42336 1/20 0.33
MINK1 Q8N4C8 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
DHFR P00374 1/20 0.33
PTGS2 P35354 1/20 0.33
KDM4E B2RXH2 5/20 0.33
CXCR4 P61073 1/20 0.33
MGLL Q99685 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TRPV4 Q9HBA0 1/20 0.31
MAT2A P31153 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17247903 0.78 LMNA (0.40) HSP90AA1HSP90AB1P2RX7KDM4ECXCR4
SCHEMBL16635491 0.78 LMNA (0.34) P2RX7KDM4ECXCR4MGLLTRPV4
SCHEMBL13260558 0.78 LMNA (0.34) P2RX7KDM4ECXCR4MGLLTRPV4
SCHEMBL29955918 0.78 MGLL (0.33) P2RX7KDM4ECXCR4MGLLTRPV4
SCHEMBL1040845 0.77 MGLL (0.32) P2RX7KDM4EMGLLHSD17B10TRPV4
SCHEMBL29951212 0.77 MGLL (0.32) P2RX7KDM4EMGLLHSD17B10TRPV4
SCHEMBL28012819 0.77 IDH1 (0.34) P2RX7KDM4EMGLLTRPV4LMNA
SCHEMBL14844546 0.74 MBOAT4 (0.36) KDM4EHSD17B10ALDH1A1KMT2A
SCHEMBL14929718 0.74
SCHEMBL17986994 0.74 HSP90AA1 (0.44) TKTHSP90AA1HSP90AB1P2RX7KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed