SCHEMBL29952853

SCHEMBL29952853

[C-]#[N+]Cc1ccc(F)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.41
DAO P14920 1/20 0.38
TSHR P16473 2/20 0.38
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
RPA1 P27694 1/20 0.36
SOS1 Q07889 1/20 0.35
PNMT P11086 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
MEN1 O00255 2/20 0.35
MAPT P10636 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CNR2 P34972 1/20 0.35
GRM4 Q14833 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29956731 0.81 HTT (0.41) DAOMEN1KMT2AALDH1A1HTT
SCHEMBL3756416 0.81 IDO1 (0.52) TSHRPNMTTAAR1MEN1MAPT
SCHEMBL29955728 0.76 CYP3A4 (0.42) PNMTMAPTALDH1A1NPSR1KDM4E
SCHEMBL29953131 0.76 KDM4E (0.44) TSHRALDH1A1NPSR1KDM4ECYP1A2
SCHEMBL318499 0.76 KDM4E (0.44) TSHRALDH1A1NPSR1KDM4ECYP1A2
SCHEMBL23850015 0.75 TAAR1 (0.47) PIK3CADAOHDAC3HDAC1HDAC2
SCHEMBL1503218 0.74 PIK3CA (0.45) PIK3CADAOTSHRHDAC3HDAC1
SCHEMBL16388285 0.74 PIK3CA (0.45) PIK3CADAOTSHRHDAC3HDAC1
SCHEMBL3538182 0.73 IDO1 (0.46) TAAR1MEN1KMT2AALDH1A1KDM4E
SCHEMBL5650950 0.72 PIK3CA (0.47) PIK3CADAOTSHRHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed