SCHEMBL29953456

SCHEMBL29953456

COc1ncc(B(O)O)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 3/20 0.40
LMNA P02545 2/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
APEX1 P27695 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAPK1 P28482 1/20 0.37
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
TTR P02766 2/20 0.35
PTGES2 Q9H7Z7 3/20 0.33
MALT1 Q9UDY8 2/20 0.33
CDK2 P24941 1/20 0.33
GSK3B P49841 1/20 0.33
KCNJ5 P48544 1/20 0.32
KCNJ3 P48549 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
PIK3CA P42336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1811195 1.00 ENPP2 (0.40) ENPP2LMNACYP2C9TSHRAPEX1
SCHEMBL14120573 0.82 RORC (0.39) ENPP2LMNACYP2C9TSHRAPEX1
SCHEMBL16734291 0.81 RORC (0.37) ENPP2LMNACYP2C9TSHRAPEX1
SCHEMBL29955039 0.80 ENPP2 (0.34) ENPP2LMNACYP2C9TSHRAPEX1
SCHEMBL24354976 0.79 ENPP2 (0.36) ENPP2CA1CA2CYP3A4MAPT
SCHEMBL3635036 0.79 ENPP2 (0.36) ENPP2CA1CA2PIK3CAMAPT
SCHEMBL20605929 0.79 PIK3CA (0.37) ENPP2CA1CA2PIK3CAMAPT
SCHEMBL29955940 0.79 ENPP2 (0.36) ENPP2CA1CA2PIK3CAMAPT
SCHEMBL366465 0.78 SCN9A (0.44) CYP2C9CYP3A4
SCHEMBL29956760 0.78 BCHE (0.38) ENPP2LMNACYP2C9TSHRAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed