SCHEMBL29954977

SCHEMBL29954977

OB(O)c1cnc2c(c1)[nH]c1cccnc12

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.46
GABRG2 P18507 2/20 0.46
GABRB3 P28472 2/20 0.46
GABRA5 P31644 2/20 0.46
GABRA3 P34903 2/20 0.46
GABRA2 P47869 2/20 0.46
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
KIF11 P52732 1/20 0.40
KCNMA1 Q12791 4/20 0.40
PARP1 P09874 3/20 0.38
DAO P14920 2/20 0.35
MAPT P10636 1/20 0.35
NUDT1 P36639 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30322789 0.76 PARP1 (0.55) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL12396542 0.76 PARP1 (0.55) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL12023644 0.73 CCR1 (0.57) MAPTKDM4E
SCHEMBL28561892 0.72 HSP90AA1 (0.40) ADORA3PARP1MAPTKDM4E
SCHEMBL20982021 0.71 AURKA (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL3719247 0.69 CA1 (0.42) MAPTKDM4E
SCHEMBL19988523 0.69 ADORA3 (0.54) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL21157142 0.69 KIF11 (0.55) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL19988521 0.67 ADORA3 (0.48) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL12590228 0.67 GABRA1 (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed