SCHEMBL29956815

SCHEMBL29956815

COc1nc(N)ncc1B(O)O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 4/20 0.43
KMT2A Q03164 1/20 0.37
P2RX3 P56373 1/20 0.36
P2RX2 Q9UBL9 1/20 0.36
CYP1A2 P05177 1/20 0.35
METAP2 P50579 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
KDR P35968 1/20 0.35
JAK3 P52333 1/20 0.35
AURKB Q96GD4 1/20 0.35
DHFR P00374 1/20 0.35
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31177244 0.78 LMNA (0.34) KMT2A
SCHEMBL25589550 0.78 LMNA (0.34) KMT2A
SCHEMBL9591 0.78 QPCT (0.37) KMT2ACYP1A2METAP2
SCHEMBL7891452 0.75 NUDT1 (0.44) NUDT1KMT2ACYP1A2METAP2AURKB
SCHEMBL29955721 0.75 DHFR (0.38) DHFR
SCHEMBL2955132 0.74 HPGD (0.38) KMT2ACYP1A2
SCHEMBL24456358 0.74 RXFP1 (0.39) NUDT1DHFR
SCHEMBL31631823 0.74 NUDT1 (0.59) NUDT1KMT2AP2RX3P2RX2CYP1A2
SCHEMBL4055122 0.74 NUDT1 (0.59) NUDT1KMT2AP2RX3P2RX2CYP1A2
SCHEMBL29956361 0.74 RXFP1 (0.39) NUDT1DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed