SCHEMBL29956882

SCHEMBL29956882

Cc1ccc(N)c(C=O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.52
ALOX15 P16050 2/20 0.52
CYP3A4 P08684 2/20 0.52
TP53 P04637 1/20 0.52
THRB P10828 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
SRC P12931 1/20 0.47
ERN1 O75460 2/20 0.46
CA1 P00915 1/20 0.45
ALDH1A1 P00352 6/20 0.44
TSHR P16473 2/20 0.44
HSD17B10 Q99714 1/20 0.41
CYP2A6 P11509 1/20 0.41
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
ALPG P10696 1/20 0.39
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3384426 1.00 TDP1 (0.52) TDP1ALOX15CYP3A4TP53THRB
P-Xylene SCHEMBL28503019 0.85 ACHE (0.46) TDP1ALOX15CYP3A4TP53THRB
SCHEMBL2888296 0.83 ERN1 (0.52) TDP1THRBSMN1; SMN2SRCERN1
SCHEMBL6257642 0.82 TDP1 (0.52) TDP1ALOX15CYP3A4TP53THRB
SCHEMBL8338685 0.77 TDP1 (0.52) TDP1ALOX15CYP3A4TP53THRB
SCHEMBL13363012 0.77 TDP1 (0.52) TDP1ALOX15CYP3A4TP53THRB
SCHEMBL268706 0.76 ALDH1A1 (0.52) TDP1SMN1; SMN2SRCERN1ALDH1A1
SCHEMBL9404722 0.76 TDP1 (0.48) TDP1ALOX15CYP3A4THRBERN1
SCHEMBL135290 0.76 TDP1 (0.40) TDP1ALOX15CYP3A4TP53THRB
SCHEMBL21507858 0.76 TDP1 (0.50) TDP1ALOX15CYP3A4TP53THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4622967-A1 COMPOUNDS THAT INHIBIT PKMYT1 Exelixis, Inc. (US) 2025-10-01 EP disclosed
WO-2024112853-A1 COMPOUNDS THAT INHIBIT PKMYT1 EXELIXIS, INC. (US) 2024-05-30 WO disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed