SCHEMBL29957029

SCHEMBL29957029

O=Cc1ccnc2[nH]c(-c3ccccc3)cc12

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.56
ADORA1 P30542 2/20 0.56
CCNB2 O95067 1/20 0.51
CDK1 P06493 1/20 0.51
CCNB1 P14635 1/20 0.51
GSK3A P49840 1/20 0.51
GSK3B P49841 1/20 0.51
CDK5 Q00535 1/20 0.51
CDK5R1 Q15078 1/20 0.51
CCNB3 Q8WWL7 1/20 0.51
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
MAPK14 Q16539 9/20 0.47
EGFR P00533 8/20 0.47
MAPKAPK2 P49137 1/20 0.43
CCR1 P32246 1/20 0.42
CCR5 P51681 1/20 0.42
CCR8 P51685 1/20 0.42
CSF1R P07333 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23624869 0.79 ADORA2A (0.54) ADORA2AADORA1CCNB2CDK1CCNB1
SCHEMBL1748962 0.77 IMPDH2 (0.47) GSK3BCDK5CDK5R1
SCHEMBL16041244 0.76 CDC7 (0.59) ADORA2AADORA1CCNB2CDK1CCNB1
SCHEMBL20928367 0.76 ADORA2A (0.56) ADORA2AADORA1CCNB2CDK1CCNB1
SCHEMBL31240593 0.76 CDC7 (0.59) ADORA2AADORA1CCNB2CDK1CCNB1
SCHEMBL1778024 0.76 ADORA2A (0.56) ADORA2AADORA1CCNB2CDK1CCNB1
SCHEMBL3604759 0.76 ADORA2A (0.56) ADORA2AADORA1CCNB2CDK1CCNB1
SCHEMBL29955037 0.76 ADORA2A (0.52) ADORA2AADORA1CCNB2CDK1CCNB1
SCHEMBL26104732 0.76 KDM5A (0.61) ADORA2AADORA1CCNB2CDK1CCNB1
SCHEMBL26102930 0.76 CDC7 (0.62) ADORA2AADORA1CCNB2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed