SCHEMBL29958253

SCHEMBL29958253

CCOC(=O)C1C(=O)Nc2cc(F)ccc2C1=O

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.50
ALDH1A1 P00352 7/20 0.42
MAPT P10636 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4E B2RXH2 3/20 0.41
TGM2 P21980 1/20 0.41
LMNA P02545 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GAA P10253 2/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
TP53 P04637 1/20 0.35
RECQL P46063 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28890594 1.00 TDP2 (0.50) TDP2ALDH1A1MAPTL3MBTL1KDM4E
SCHEMBL9201592 0.85 TDP2 (0.50) TDP2ALDH1A1MAPTL3MBTL1KDM4E
SCHEMBL28087596 0.81 ALDH1A1 (0.56) TDP2ALDH1A1MAPTL3MBTL1KDM4E
SCHEMBL9204538 0.81 TDP2 (0.46) TDP2ALDH1A1MAPTLMNAMEN1
SCHEMBL15313181 0.80 TDP2 (0.43) TDP2ALDH1A1MAPTL3MBTL1KDM4E
SCHEMBL13295304 0.79 TDP2 (0.49) TDP2ALDH1A1MAPTL3MBTL1KDM4E
SCHEMBL28890601 0.78 TDP2 (0.40) TDP2ALDH1A1MAPTL3MBTL1KDM4E
SCHEMBL2776008 0.75 KDM4E (0.42) TDP2ALDH1A1MAPTL3MBTL1KDM4E
SCHEMBL9705021 0.75 KDM4E (0.42) TDP2ALDH1A1MAPTL3MBTL1KDM4E
SCHEMBL9204906 0.75 TDP2 (0.40) TDP2ALDH1A1HPGDTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115362155-B Arylamine derivative, preparation method and medical application thereof 中国医药研究开发中心有限公司 2024-06-18 CN disclosed
CN-115362155-A Arylamine derivatives, and preparation method and medical application thereof 中国医药研究开发中心有限公司 2022-11-18 CN disclosed