SCHEMBL29960805

SCHEMBL29960805

O=C(NCC1CCN(Cc2ccc(F)cc2)CC1)c1cccnc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 3/20 0.67
ACHE P22303 1/20 0.59
GSK3B P49841 1/20 0.59
LMNA P02545 1/20 0.57
HDAC3 O15379 3/20 0.55
HDAC4 P56524 3/20 0.55
HDAC1 Q13547 3/20 0.55
HDAC7 Q8WUI4 3/20 0.55
HDAC2 Q92769 3/20 0.55
HDAC10 Q969S8 3/20 0.55
HDAC11 Q96DB2 3/20 0.55
HDAC8 Q9BY41 3/20 0.55
HDAC6 Q9UBN7 3/20 0.55
HDAC9 Q9UKV0 3/20 0.55
HDAC5 Q9UQL6 3/20 0.55
CCR2 P41597 2/20 0.53
KCNH2 Q12809 2/20 0.53
CHRM4 P08173 1/20 0.53
HTR4 Q13639 2/20 0.51
MEN1 O00255 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29960884 0.89 CACNA1I (0.66) CACNA1IACHEGSK3BHDAC3HDAC4
SCHEMBL29960540 0.89 CACNA1I (0.66) CACNA1IACHEGSK3BHDAC3HDAC4
SCHEMBL29280913 0.86 CACNA1I (0.52) CACNA1IACHEGSK3BKCNH2KMT2A
SCHEMBL29960822 0.84 ACHE (0.62) CACNA1IACHEGSK3BHDAC3HDAC4
SCHEMBL29960939 0.82 CACNA1I (0.66) CACNA1IGSK3BLMNAHDAC3HDAC4
Trifluoroacetic Acid SCHEMBL29280901 0.81 CACNA1I (0.48) CACNA1IACHEGSK3BHDAC3HDAC4
SCHEMBL5368811 0.81 HDAC3 (0.64) CACNA1ILMNAHDAC3HDAC4HDAC1
SCHEMBL29960926 0.80 GSK3B (0.64) CACNA1IACHEGSK3BHDAC3HDAC4
SCHEMBL29961434 0.80 FABP6 (0.62) CACNA1IACHEGSK3BLMNAHDAC3
SCHEMBL22583343 0.80 THRB (0.64) CACNA1IHDAC1HDAC6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112047928-B Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2022-09-23 CN claimed
CN-112047928-B Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2022-09-23 CN disclosed