SCHEMBL29960939

SCHEMBL29960939

Cc1cccc(CN2CCC(CNC(=O)c3cccnc3)CC2)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 2/20 0.66
GSK3B P49841 1/20 0.62
CCR2 P41597 1/20 0.58
HDAC3 O15379 4/20 0.58
HDAC4 P56524 4/20 0.58
HDAC1 Q13547 4/20 0.58
HDAC7 Q8WUI4 4/20 0.58
HDAC2 Q92769 4/20 0.58
HDAC10 Q969S8 4/20 0.58
HDAC11 Q96DB2 4/20 0.58
HDAC8 Q9BY41 4/20 0.58
HDAC6 Q9UBN7 4/20 0.58
HDAC9 Q9UKV0 4/20 0.58
HDAC5 Q9UQL6 4/20 0.58
ACKR3 P25106 2/20 0.55
KCNH2 Q12809 1/20 0.55
KMT2A Q03164 1/20 0.54
HTR4 Q13639 1/20 0.54
TSHR P16473 2/20 0.53
USP2 O75604 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29960540 0.88 CACNA1I (0.66) CACNA1IGSK3BHDAC3HDAC4HDAC1
SCHEMBL29960926 0.87 GSK3B (0.64) CACNA1IGSK3BHDAC3HDAC4HDAC1
SCHEMBL29960884 0.84 CACNA1I (0.66) CACNA1IGSK3BCCR2HDAC3HDAC4
SCHEMBL29960805 0.82 CACNA1I (0.67) CACNA1IGSK3BCCR2HDAC3HDAC4
SCHEMBL29961434 0.82 FABP6 (0.62) CACNA1IGSK3BHDAC3HDAC4HDAC1
SCHEMBL23013174 0.78 CACNA1I (0.69) CACNA1IGSK3BHDAC3HDAC4HDAC1
SCHEMBL28905792 0.78 GSK3B (1.00) GSK3BACKR3
SCHEMBL28361465 0.78 CCR2 (0.55) CACNA1IGSK3BCCR2HDAC3HDAC4
SCHEMBL29960822 0.78 ACHE (0.62) CACNA1IGSK3BHDAC3HDAC4HDAC1
SCHEMBL22583343 0.78 THRB (0.64) CACNA1IHDAC1HDAC6KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112047928-B Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2022-09-23 CN claimed
CN-112047928-B Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2022-09-23 CN disclosed