SCHEMBL299609

SCHEMBL299609

CC(c1cc(C(F)(F)F)nn1Oc1ccccn1)C(C(N)=O)c1ccc2[nH]ccc2c1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.36
PTGS2 P35354 1/20 0.34
CTNNB1 P35222 2/20 0.33
WNT3A P56704 2/20 0.33
FYN P06241 1/20 0.33
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
SYK P43405 1/20 0.31
CHRNA7 P36544 1/20 0.30
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
SRPK1 Q96SB4 1/20 0.30
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL299138 0.86 PTGS2 (0.35) NR3C1PTGS2SYKCHRNA7CYP19A1
SCHEMBL299025 0.78 TRPV1 (0.46)
SCHEMBL297590 0.66 TRPV1 (0.56)
SCHEMBL299097 0.64 TRPV1 (0.44)
SCHEMBL30795530 0.60 PTGS2 (0.49) NR3C1PTGS2CTNNB1WNT3ASLC6A2
SCHEMBL3428521 0.59 NPC1 (0.56) PTGS2CTNNB1WNT3ASLC6A2SLC6A4
SCHEMBL5496056 0.59 SLC6A2 (0.55) NR3C1PTGS2CTNNB1WNT3AFYN
SCHEMBL6263511 0.58 PTGS2 (0.78) PTGS2SLC6A2SLC6A4SLC6A3
SCHEMBL8869741 0.58 PDE10A (0.44) PTGS2CTNNB1WNT3ASLC6A2SLC6A4
SCHEMBL3425528 0.57 ABL1 (0.42) NR3C1PTGS2SYKCHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427436-A1 SUBSTITUTED AROMATIC CARBOXAMIDE AND UREA DERIVATIVES AS VANILLOID RECEPTOR LIGANDS Grünenthal GmbH (DE) 2012-03-14 EP claimed
WO-2010127855-A1 SUBSTITUTED AROMATIC CARBOXAMIDE AND UREA DERIVATIVES AS VANILLOID RECEPTOR LIGANDS Grünenthal GmbH (DE) 2010-11-11 WO claimed