SCHEMBL8869741

SCHEMBL8869741

c1ccc(Oc2ccc3[nH]ccc3c2)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.44
CTNNB1 P35222 1/20 0.44
WNT3A P56704 1/20 0.44
KDR P35968 1/20 0.44
PRKCQ Q04759 1/20 0.44
NPC1 O15118 1/20 0.42
TLR4 O00206 1/20 0.42
TLR2 O60603 1/20 0.42
KDM4E B2RXH2 1/20 0.42
LTA4H P09960 1/20 0.42
MAP4K4 O95819 1/20 0.41
SCN7A Q01118 4/20 0.40
KCNH2 Q12809 4/20 0.40
HRH3 Q9Y5N1 1/20 0.40
CYP2D6 P10635 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
PTGS2 P35354 1/20 0.39
DHODH Q02127 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8870430 0.83 RAB9A (0.54) CTNNB1WNT3AKDRPRKCQNPC1
SCHEMBL13548670 0.78 ALDH1A1 (0.45) KDRPRKCQNPC1KDM4ELTA4H
SCHEMBL2509875 0.78 AHR (0.45) KDRPRKCQLTA4HAHR
SCHEMBL962086 0.78 L3MBTL1 (0.46) KDRPRKCQNPC1LTA4HPTGS2
SCHEMBL443361 0.77 NPC1 (0.55) PRKCQNPC1LTA4HTRPA1CA1
SCHEMBL2778800 0.77 KDR (0.50) KDRPRKCQLTA4HAHR
SCHEMBL2434619 0.77 KDR (0.45) KDRPRKCQLTA4HAHR
SCHEMBL13548673 0.77 CYP3A4 (0.47) PDE10AKDRPRKCQNPC1LTA4H
SCHEMBL18756060 0.77 KDR (0.42) KDRPRKCQLTA4HAHR
SCHEMBL18392981 0.77 MAPT (0.52) PDE10ACTNNB1WNT3ANPC1TLR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637593-A MIGRAINE; HYPOTENSIVE AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-06-10 US disclosed
EP-0674619-A1 TRYPTAMINE ANALOGUES AS 5-HT 1?-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-10-04 EP disclosed
WO-1994014770-A1 TRYPTAMINE ANALOGUES AS 5-HT1-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-07-07 WO disclosed