SCHEMBL29962149

SCHEMBL29962149

CNC(=O)N1CCc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.52
HTR2C P28335 1/20 0.50
ATM Q13315 1/20 0.47
LMNA P02545 2/20 0.46
NPC1 O15118 2/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
ADRB2 P07550 1/20 0.46
ADRB1 P08588 1/20 0.46
ADRB3 P13945 1/20 0.46
ROCK1 Q13464 1/20 0.44
NOTUM Q6P988 1/20 0.43
CREBBP Q92793 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
DRD4 P21917 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.41
MEN1 O00255 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2845681 0.89 HTR2C (0.61) HTR2CATMLMNANPC1MAPT
SCHEMBL981641 0.85 NOTUM (0.60) DRD2LMNANPC1MAPTHTT
SCHEMBL27872558 0.84 DRD2 (0.57) DRD2HTR2CATMLMNANPC1
SCHEMBL29962960 0.84 DRD2 (0.52) DRD2HTR2CLMNANPC1MAPT
SCHEMBL3318846 0.84 DRD2 (0.52) DRD2HTR2CLMNANPC1MAPT
SCHEMBL3735431 0.83 DRD2 (0.56) DRD2HTR2CATMLMNANPC1
SCHEMBL2851575 0.82 RAB9A (0.64) DRD2HTR2CATMNPC1MAPT
SCHEMBL7754766 0.81 DRD2 (0.55) DRD2HTR2CLMNANPC1MAPT
SCHEMBL7267829 0.79 DRD2 (0.44) DRD2HTR2CATMNPC1RAB9A
SCHEMBL2203452 0.79 DRD2 (0.58) DRD2LMNANPC1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115141179-B Novel benzoheterocyclyl derivative, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2024-09-13 CN disclosed
CN-115141179-A Novel benzo heterocyclic derivatives, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-10-04 CN disclosed