SCHEMBL29965486

SCHEMBL29965486

O=C(O)c1nc2ccccc2c(=O)[nH]1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 2/20 0.58
TOP2B Q02880 2/20 0.58
BRD4 O60885 1/20 0.58
PARP1 P09874 4/20 0.58
TNKS2 Q9H2K2 4/20 0.58
QTRT1 Q9BXR0 1/20 0.58
TNKS O95271 2/20 0.56
PARP2 Q9UGN5 1/20 0.55
PKM P14618 1/20 0.53
GUSB P08236 2/20 0.53
KDM4E B2RXH2 2/20 0.53
HPGD P15428 1/20 0.53
KMT2A Q03164 4/20 0.52
MEN1 O00255 3/20 0.52
ATM Q13315 1/20 0.52
MAPT P10636 2/20 0.52
MAPK1 P28482 1/20 0.51
ALDH1A1 P00352 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
TP53 P04637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4936991 1.00 TOP2A (0.58) TOP2ATOP2BBRD4PARP1TNKS2
SCHEMBL28060714 0.86 BRD4 (0.59) TOP2ATOP2BBRD4PARP1TNKS2
SCHEMBL941961 0.86 QTRT1 (0.59) TOP2ATOP2BBRD4PARP1TNKS2
SCHEMBL27334538 0.84 BRD4 (0.74) TOP2ATOP2BBRD4PARP1TNKS2
SCHEMBL8187460 0.84 TOP2A (0.59) TOP2ATOP2BBRD4PARP1TNKS2
SCHEMBL11548593 0.83 KDM4E (0.59) TOP2ATOP2BBRD4PARP1TNKS2
SCHEMBL28851317 0.82 TOP2A (0.44) TOP2ATOP2BBRD4PARP1TNKS2
SCHEMBL942595 0.82 MAPT (0.56) TOP2ATOP2BBRD4PARP1TNKS2
SCHEMBL6157123 0.82 MAPT (0.56) TOP2ATOP2BBRD4PARP1TNKS2
SCHEMBL11499700 0.82 TOP2A (0.52) TOP2ATOP2BBRD4PARP1TNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115109050-A Preparation method and application of quinazolinone-based 1,3, 4-oxadiazole compound 天津理工大学 2022-09-27 CN claimed
CN-117384156-B Preparation method and application of camelning alkali A and derivative thereof 烟台大学 2024-03-15 CN disclosed
CN-117384156-A Preparation method and application of camelning alkali A and derivative thereof 烟台大学 2024-01-12 CN disclosed
CN-115109050-A Preparation method and application of quinazolinone-based 1,3, 4-oxadiazole compound 天津理工大学 2022-09-27 CN disclosed